Search Count: 10
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Crystals Structure Of B-Raf Kinase Domain In Complex With An Imidazopyridinyl Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2017-11-22 Classification: Transferase/Transferase Inhibitor Ligands: 8EN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-22
Ligands: 8EN
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P38 Alpha Mutant C162S In Complex With Cmpd2 [N-(4-Methyl-3-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Phenyl)-3-(Trifluoromethyl)Benzamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2017-11-15 Classification: TRANSFERASE Ligands: 8EN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-15
Ligands: 8EN
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Discovery Of Imidazo[1,2-A]-Pyridine Inhibitors Of Pan-Pi3 Kinases That Are Efficacious In A Mouse Xenograft Model
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 5XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: GOL, 5XV
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Identification Of N-(4-((1R,3S,5S)-3-Amino-5-Methylcyclohexyl)Pyridin-3-Yl)-6-(2,6-Difluorophenyl)-5-Fluoropicolinamide (Pim447), A Potent And Selective Proviral Insertion Site Of Moloney Murine Leukemia (Pim) 1,2 And 3 Kinase Inhibitor In Clinical Trials For Hematological Malignancies
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-11-11 Classification: Transferase/Transferase Inhibitor Ligands: 5H7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: 5H7
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Pim1 Complexed With A Phenylcarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2HV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: 2HV
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Pim1 Complexed With A Pyridylcarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2HW, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: 2HW, GOL
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Pim1 Complexed With A Pyridylcarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2HX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: 2HX
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Structure Of Pi3K Gamma With Imidazopyridine Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2013-07-17 Classification: Transferase/Transferase Inhibitor Ligands: 1UJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: 1UJ, SO4
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Structure Of Pi3K Gamma With Imidazopyridine Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2013-07-17 Classification: Transferase/Transferase Inhibitor Ligands: 1UK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: 1UK, SO4
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Crystal Structure Of Pi3K Gamma With N6-(3,4-Dimethoxyphenyl)-2-Morpholino-[4,5'-Bipyrimidine]-2',6-Diamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-08-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 13K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: 13K, SO4