Search Count: 52
![]() |
Crystal Structure Of The Hpk1 Kinase Domain In Complex With Inhibitor 5B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2026-08-05 Classification: TRANSFERASE Ligands: A1KCT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1KCT, EDO
![]() |
Crystal Structure Of The Hpk1 Kinase Domain In Complex With Inhibitor 6B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2026-08-05 Classification: TRANSFERASE Ligands: A1KCQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1KCQ, EDO
![]() |
Crystal Structure Of The Hpk1 Kinase Domain In Complex With Inhibitor 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2026-08-05 Classification: TRANSFERASE Ligands: A1KCR, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1KCR, EDO
![]() |
Crystal Structure Of Hpk1 T165E/S171E In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITC
![]() |
Crystal Structure Of Hpk1 T165E/S171E In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITA
![]() |
Crystal Structure Of Hpk1 T165E/S171E In Complex With Pyrazine Carboxamide Inhibitor Az3246 (Compound 24)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITB, EDO
![]() |
E3 Ligase Cbl-B In Complex With A Triazolone Core Inhibitor (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IEW, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IEW, ZN, NA
![]() |
E3 Ligase Cbl-B In Complex With A Lactam Scaffold Inhibitor (Compound 7)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IEV, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IEV, ZN, NA
![]() |
E3 Ligase Cbl-B In Complex With A Carbamate Scaffold Inhibitor (Compound 12)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IE5, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IE5, ZN, NA
![]() |
Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 31)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2024-01-24 Classification: LIGASE Ligands: ZN, NA, WX9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-24
Ligands: ZN, NA, WX9
![]() |
Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: WUQ, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: WUQ, ZN, NA
![]() |
Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: WX0, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: WX0, ZN, NA
![]() |
Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 30)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: ZN, NA, WUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: ZN, NA, WUI
![]() |
Estrogen Receptor Alpha In Complex With Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2023-02-01 Classification: TRANSCRIPTION Ligands: H09 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: H09
![]() |
Oestrogen Receptor Ligand Binding Domain In Complex With Compound 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-02-01 Classification: GENE REGULATION Ligands: GZI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: GZI
![]() |
Crystal Structure Of At7 In Complex With The Second Bromodomain Of Human Brd4 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IZR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IZR
![]() |
Crystal Structure Of The Bromodomain Of Atad2 With Az13824374
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 96L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 96L
![]() |
Crystal Structure Of The Bromodomain Of Atad2 With Phenol Hts Hit (Cpd 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 963 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 963
![]() |
Crystal Structure Of The Bromodomain Of Atad2 With Triazolopyridine (Cpd 14)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 95O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 95O
![]() |
Crystal Structure Of The Bromodomain Of Atad2 With Triazolopyridazine (Cpd 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 93L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 93L
