Search Count: 14
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Structure Of Cbl-B Bound To Compound 33
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2026-07-01 Classification: LIGASE Ligands: GOL, IOD, EDO, MG, ZN, A1DCD, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: GOL, IOD, EDO, MG, ZN, A1DCD, DMS
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Structure Of C-Cbl Bound To Compound 33
Organism: Schistosoma japonicum, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2026-07-01 Classification: LIGASE Ligands: A1DCD, ZN, MG |
Organism: Schistosoma japonicum, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: A1DCD, ZN, MG
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Structure Of Cbl-B Bound To Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2026-07-01 Classification: LIGASE/INHIBITOR Ligands: GOL, ZN, EDO, MG, A1DCC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: GOL, ZN, EDO, MG, A1DCC
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Crystal Structure Of Cbl-B Tkb Bound To Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2024-07-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, A1AEG, GOL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MG, A1AEG, GOL, PEG
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Crystal Structure Of Cbl-B Tkb Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2024-07-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, CA, A1AD4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MG, CA, A1AD4
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Crystal Structure Of Braf In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: V5J, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: V5J, IOD
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Crystal Structure Of Braf In Complex With Inhibitor Gne-0749
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: VQP, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: VQP, CL
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Human Immunoproteasome 20S Particle In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2019-09-11 Classification: HYDROLASE Ligands: SCN, NA, HUJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-11
Ligands: SCN, NA, HUJ
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Synthesis, Characterization And Pk/Pd Studies Of A Series Of Spirocyclic Pyranochromene Bace1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-05-14 Classification: Hydrolase/Hydrolase inhibitor Ligands: NI, 2X4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-14
Ligands: NI, 2X4
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Synthesis, Characterization And Pk/Pd Studies Of A Series Of Spirocyclic Pyranochromene Bace1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-05-14 Classification: hydrolase/hydrolase inhibitor Ligands: NI, 2X5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-14
Ligands: NI, 2X5
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Diethylaminosulfur Trifluoride-Mediated Intramolecular Cyclization Of 2-Hydroxy-Benzylureas To Fused Bicyclic Aminooxazoline Compounds And Evaluation Of Their Biochemical Activity Against Beta-Secretase-1 (Bace1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2013-09-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1W0, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: 1W0, DMS
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Diethylaminosulfur Trifluoride-Mediated Intramolecular Cyclization Of 2-Hydroxy-Benzylureas To Fused Bicyclic Aminooxazoline Compounds And Evaluation Of Their Biochemical Activity Against Beta-Secretase-1 (Bace-1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-09-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1W1, ACT, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: 1W1, ACT, DMS
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Diethylaminosulfur Trifluoride-Mediated Intramolecular Cyclization Of 2-Hydroxy-Benzylureas To Fused Bicyclic Aminooxazoline Compounds And Evaluation Of Their Biochemical Activity Against Beta-Secretase-1 (Bace-1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2013-09-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1W2, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: 1W2, ACT
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Aminooxazoline Inhibitor Of Bace-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-09-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NI, 1WP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: NI, 1WP
