Search Count: 9
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Fgfr2 Kinase Domain Bound To Reversible Inhibitor Cmpd 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2024-02-14 Classification: ONCOPROTEIN Ligands: GOL, GSH, WXQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: GOL, GSH, WXQ
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Fgfr2 Kinase Domain Bound To Irreversible Inhibitor Cmpd 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.33 Å Release Date: 2024-02-14 Classification: Transferase/Inhibitor Ligands: GOL, UIM, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: GOL, UIM, SO4
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Discovery And Clinical Validation Of Rly-4008, The First Highly Selective Fgfr2 Inhibitor With Activity Across Fgfr2 Alterations And Resistance Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.79 Å Release Date: 2023-06-07 Classification: TRANSFERASE/INHIBITOR Ligands: WCJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: WCJ
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A Multiconformer Ligand Model Of Ek6 Bound To Erk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2018-12-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, EDO, EK6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: SO4, EDO, EK6
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A Multiconformer Ligand Model Of Acylenzyme Intermediate Of Meropenem Bound To An Sfc-1 E166A Mutant
Organism: Serratia fonticola
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-12-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: EDO, MER |
Organism: Serratia fonticola
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: EDO, MER
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A Multiconformer Ligand Model Of 5T5 Bound To Bace-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-12-19 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
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A Multiconformer Ligand Model Of Inhibitor 53W Bound To Creb Binding Protein Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2018-12-19 Classification: transcription/transcription inhibitor Ligands: 53W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: 53W
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A Multiconformer Ligand Model Of An Isoxazolyl-Benzimidazole Ligand Bound To The Bromodomain Of Human Crebbp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-12-19 Classification: transcription/transcription inhibitor Ligands: NO3, 2LL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: NO3, 2LL, EDO
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A Multiconformer Ligand Model Of 3,5 Dimethylisoxaxole Bound To The Bromodomain Of Human Brd4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2018-12-19 Classification: transcription/transcription inhibitor Ligands: EDO, 9BM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: EDO, 9BM