Search Count: 8
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Wd Repeat-Containing Protein 5 Complexed With 4-(7-((1H-Imidazol-1-Yl)Methyl)-5-(1-Methyl-3-(Trifluoromethyl)-1H-Pyrazol-4-Yl)-1-Oxo-3,4-Dihydroisoquinolin-2(1H)-Yl)-6-Ethyl-N-Methylquinoline-8-Carboxamide (Compound 10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2023-01-11 Classification: TRANSCRIPTION Ligands: BEN, UY9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-11
Ligands: BEN, UY9
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Wdr5 In Complex With A Win Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-03-13 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HH7, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HH7, DMS, SO4
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Wdr5 In Complex With A Win Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2019-03-13 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HHM, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HHM, SO4, DMS
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Discovery Of Potent 2-Aryl-6,7-Dihydro-5Hpyrrolo[ 1,2-A]Imidazoles As Wdr5 Win-Site Inhibitors Using Fragment-Based Methods And Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLM
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLP
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLS, SO4
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLJ, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLJ, EPE
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Crystal Structure Of Wdr5 In Complex With Myc Mbiiib Peptide
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-04-15 Classification: DNA BINDING PROTEIN Ligands: TRS, EDO |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2015-04-15
Ligands: TRS, EDO