Search Count: 22
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Tnni3K Complexed With N-Methyl-4-(4-(3-(3-(Trifluoromethyl) Phenyl) Ureido) Phenoxy)Picolinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2021-11-10 Classification: TRANSFERASE/INHIBITOR Ligands: ZFS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: ZFS
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Tnni3K Complexed With 1-(3,5-Dichloro-4-((6-(Methylamino)Pyrimidin-4-Yl)Oxy)Phenyl)-3-(3-(Trifluoromethyl)Phenyl)Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2021-11-10 Classification: TRANSFERASE/INHIBITOR Ligands: ZGD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: ZGD
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Bmp1 Complexed With A Reverse Hydroxymate - Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-08-08 Classification: HYDROLASE Ligands: SCN, ZN, EVV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SCN, ZN, EVV, EDO
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Bmp1 Complexed With A Reverse Hydroxamate - Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2018-08-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, E7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: ZN, E7D
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Bmp1 Complexed With A Reverse Hydroxymate - Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-08-08 Classification: HYDROLASE Ligands: EDO, ZN, E8M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: EDO, ZN, E8M
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Bmp1 Complexed With (2~{S})-2-[[(1~{R},3~{S},4~{S})-2-[(2~{R})-2-[2-(Oxidanylamino)-2-Oxidanylidene-Ethyl]Heptanoyl]-2-Azabicyclo[2.2.1]Heptan-3-Yl]Carbonylamino]-2-Phenyl-Ethanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-08-08 Classification: HYDROLASE Ligands: SCN, ZN, E8P, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SCN, ZN, E8P, EDO
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Bmp1 Complexed With A Hydroxamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2018-08-08 Classification: HYDROLASE Ligands: SCN, ZN, E8J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SCN, ZN, E8J
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Bmp1 Complexed With A Hydroxamate - Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2018-08-08 Classification: HYDROLASE Ligands: SCN, ZN, E8S, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SCN, ZN, E8S, EDO
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Tnni3K Complexed With A 4,6-Diaminopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.97 Å Release Date: 2018-04-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CV4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: CV4
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Crystal Structure Of Human Renin In Complex With A Biphenylpipderidinylcarbinol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 90D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, 90D
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Crystal Structure Of Human Renin In Complex With A Biphenylpipderidinylcarbinol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 9G7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, 9G7, SO4
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Crystal Structure Of Human Renin In Complex With A Biphenylpipderidinylcarbinol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, SO4, 9JD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, SO4, 9JD
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Braf Complexed With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2016-03-16 Classification: Transferase/Transferase Inhibitor Ligands: GOL, 4EF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-16
Ligands: GOL, 4EF
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Tnni3K Complexed With Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.07 Å Release Date: 2015-09-23 Classification: Transferase/Transferase Inhibitor Ligands: 4CV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-23
Ligands: 4CV
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Tnni3K Complexed With Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-09-23 Classification: Transferase/Transferase Inhibitor Ligands: 4CW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-23
Ligands: 4CW
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Soluble Epoxide Hydrolase Complexed With A Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2013-06-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 1LF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: 1LF
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Co-Crystal Structure Of Checkpoint Kinase Chk1 With A Pyrrolo-Pyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2006-06-13 Classification: SIGNALING PROTEIN, TRANSFERASE Ligands: SO4, 199 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: SO4, 199
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Fk506 Binding Protein Mutant, Homodimeric Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2000-08-09 Classification: ISOMERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2000-08-09
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Fkbp Mutant F36V Complexed With Remodeled Synthetic Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 1998-09-02 Classification: ISOMERASE Ligands: AP1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1998-09-02
Ligands: AP1
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Design, Synthesis, And Kinetic Evaluation Of High-Affinity Fkbp Ligands, And The X-Ray Crystal Structures Of Their Complexes With Fkbp12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1994-01-31 Classification: CIS-TRANS ISOMERASE Ligands: SB3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1994-01-31
Ligands: SB3
