Search Count: 20
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Structural Basis And Sar For Od 270, A Lead Stage 1,2,4-Triazole Based Specific Tankyrase1/2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2013-03-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: NCA, ZN, 1AK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: NCA, ZN, 1AK
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Crystal Structure Of Human Renin Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2006-12-05 Classification: HYDROLASE Ligands: LIY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-12-05
Ligands: LIY
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Crystal Structure Of Human Renin Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2006-12-05 Classification: HYDROLASE Ligands: LIX, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-12-05
Ligands: LIX, CIT
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Crystal Structure Of Human Renin Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-11-14 Classification: HYDROLASE Ligands: 7IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-14
Ligands: 7IG
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Human Renin/Pf02342674 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2006-10-24 Classification: HYDROLASE Ligands: UA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-10-24
Ligands: UA4
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The C Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-06-20 Classification: HYDROLASE Ligands: L1A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-20
Ligands: L1A
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The C Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: PZ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: PZ1
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 1IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 1IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 2IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 2IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The C Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 3IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 3IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The C Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 4IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 4IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 5IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 5IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: L1B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: L1B
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: NAG, 6IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: NAG, 6IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: 7IG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: 7IG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: 3LG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: 3LG
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Ketopiperazine-Based Renin Inhibitors: Optimization Of The "C" Ring
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2006-06-13 Classification: HYDROLASE Ligands: 4LG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-13
Ligands: 4LG
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Crystal Structure Of Renin-Pf00074777 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2006-04-05 Classification: HYDROLASE Ligands: PZ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-04-05
Ligands: PZ1
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Crystal Structure Of Renin-Pf00257567 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2006-04-05 Classification: HYDROLASE Ligands: RPF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-04-05
Ligands: RPF
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Crystal Structure Of Ptp1B Complexed With 7-(1,1-Dioxo-1H-Benzo[D]Isothiazol-3-Yloxymethyl)-2-(Oxalyl-Amino)-4,7-Dihydro-5H-Thieno[2,3-C]Pyran-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2002-05-08 Classification: HYDROLASE Ligands: DBD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-05-08
Ligands: DBD
