Search Count: 11
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Identification Of Lxrbeta Selective Agonists For The Treatment Of Alzheimer'S Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-04-06 Classification: SIGNALING PROTEIN Ligands: 668, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: 668, PEG
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Identification Of Lxrbeta Selective Agonists For The Treatment Of Alzheimer'S Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2016-04-06 Classification: SIGNALING PROTEIN Ligands: 668, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: 668, SO4
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Pde10 Complexed With 4-Isopropoxy-2-(2-(3-(4-Methoxyphenyl)-4-Oxo-3,4-Dihydroquinazolin-2-Yl)Ethyl)Isoindoline-1,3-Dione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-08-12 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, MG, 4PX, 4Q0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: ZN, MG, 4PX, 4Q0
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Bace1 In Complex With 4-(Cyclohexylamino)-1-(3-Fluorophenyl)-8-(3-Isopropoxybenzyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QA
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Bace1 In Complex With 8-(3-((1-Aminopropan-2-Yl)Oxy)Benzyl)-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-08-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: 4QD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QD
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Bace1 In Complex With 8-Benzyl-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-7-Methyl-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QF
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Thrombin In Complex With An Azafluorenyl Inhibitor 23B
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2005-06-07 Classification: BLOOD CLOTTING,HYDROLASE/INHIBITOR Ligands: 062 |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-06-07
Ligands: 062
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Crystal Structure Of Thrombin In Complex With Compound 1
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2004-06-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 176 |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2004-06-08
Ligands: 176
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Crystal Structure Of Thrombin In Complex With Compound 14B
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2004-06-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 177 |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2004-06-08
Ligands: 177
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Crystal Structure Of Thrombin In Complex With L-378,622
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2004-04-06 Classification: BLOOD CLOTTING,HYDROLASE/INHIBITOR Ligands: CDA |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-04-06
Ligands: CDA
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Thrombin-Hirugen_L-378,650
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2004-04-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CDB |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-04-06
Ligands: CDB
