Search Count: 23
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Cryoem Structure Of Activated Craf/Mek/14-3-3 Complex With Nst-628
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-17
Ligands: A1AHE
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Activated Craf/Mek Heterotetramer From Focused Refinement Of Craf/Mek/14-3-3 Complex
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-17
Ligands: A1AHE
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Crystal Structure Of Ksr1/Mek1 Complex Heterotetramer With Nst-628
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE, ANP, MG, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: A1AHE, ANP, MG, EDO, CL
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Crystal Structure Of Araf/Mek1 Complex With Nst-628 And A Raf Dimer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE, MG, ANP, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: A1AHE, MG, ANP, EDO, GOL
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Crystal Structure Of Braf/Mek1 Complex With Nst-628 And An Active Raf Dimer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE, ANP, MG, EDO, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: A1AHE, ANP, MG, EDO, TRS
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Crystal Structure Of Braf/Mek Complex With Nst-628 And Inactive Raf
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: ANP, MG, A1AHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: ANP, MG, A1AHE
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Crystal Structure Of Craf/Mek1 Complex With Nst-628 And Inactive Raf
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: ANP, MG, NI, ACT, EDO, A1AHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: ANP, MG, NI, ACT, EDO, A1AHE
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Crystal Structure Of Craf/Mek Complex With Nst-628 And Active Raf Dimer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2024-04-17 Classification: TRANSFERASE Ligands: A1AHE, ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-17
Ligands: A1AHE, ANP, MG
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P21-Activated Kinase 1 In Complex With A 4-Azaindole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2017-10-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: C7Y, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: C7Y, SO4
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Crystal Structure Of P21-Activated Kinase 1 (Pak1) In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6BZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 6BZ
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound G-5555
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59T
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound Frax1036
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59U, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59U, DMS
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Crystal Structure Of P21 Activated Kinase 1 In Complex With An Inhibitor Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-07-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4T3, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: 4T3, SO4, DMS
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Crystal Structure Of P21-Activated Kinase 1 In Complex With An Inhibitor Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-07-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4T5, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: 4T5, SO4, DMS
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Crystal Structure Of P21-Activated Kinase 1 In Complex With An Inhibitor Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2015-07-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4T6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: 4T6, SO4
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Crystal Structure Of P21-Activated Kinase 4 In Complex With An Inhibitor Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-07-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4T6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: 4T6
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 7KC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 7KC
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OL
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OL
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Back Pocket Flexibility Provides Group-Ii Pak Selectivity For Type 1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2014-02-12 Classification: transferase/transferase inhibitor Ligands: 2OQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2OQ
