Search Count: 17
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Crystal Structure Of Human Clk1 Kinase In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-11-06 Classification: SIGNALING PROTEIN Ligands: SO4, XQX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: SO4, XQX
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Crystal Structure Of Human Acvr1 (Alk2) Kinase In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2024-11-06 Classification: SIGNALING PROTEIN Ligands: SO4, XQX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: SO4, XQX
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Structure Of Human Bruton'S Tyrosine Kinase In Complex With Evobrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2019-08-14 Classification: Transferase/Transferase Inhibitor Ligands: CL, MZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: CL, MZJ
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Crystal Structure Of Fgfr4 With An Irreversible Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2015-04-01 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 40M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-01
Ligands: SO4, 40M
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Crystal Structure Of Benzamide 9 Bound To Auroraa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-08-18 Classification: TRANSFERASE Ligands: LJE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-18
Ligands: LJE
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Crystal Structure Of Anthranilamide 10 Bound To Auroraa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2010-08-18 Classification: TRANSFERASE Ligands: LJF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-18
Ligands: LJF
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Pyridyl-Pyrimidine Benzimidazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2009-08-25 Classification: TRANSFERASE Ligands: K11, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-08-25
Ligands: K11, EDO
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Crystal Structure Of Human Jnk3 Complexed With N-(3-Methyl-4-(3-(2-(Methylamino)Pyrimidin-4-Yl)Pyridin-2-Yloxy)Naphthalen-1-Yl)-1H-Benzo[D]Imidazol-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-01-06 Classification: TRANSFERASE Ligands: BZ9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-06
Ligands: BZ9
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Structure Of Auroraa With Pyridyl-Pyrimidine Urea Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2008-12-23 Classification: Transferase/Inhibitor Ligands: AK8, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-23
Ligands: AK8, SO4
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Crystal Structure Of Pyrimidine Amide 11 Bound To Lck
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2007-12-18 Classification: TRANSFERASE Ligands: 9NH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-18
Ligands: 9NH
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Synthesis, Structural Analysis, And Sar Studies Of Triazine Derivatives As Potent, Selective Tie-2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-03-20 Classification: TRANSFERASE Ligands: RAJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: RAJ
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Synthesis, Structural Analysis, And Sar Studies Of Triazine Derivatives As Potent, Selective Tie-2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2007-03-20 Classification: TRANSFERASE Ligands: MUH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: MUH
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Pyridinyl-Triazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2007-03-20 Classification: TRANSFERASE Ligands: 994 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: 994
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Nicotinamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-03-20 Classification: TRANSFERASE Ligands: 608 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: 608
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Evolution Of A Highly Selective And Potent 2-(Pyridin-2-Yl)-1,3,5-Triazine Tie-2 Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-03-20 Classification: TRANSFERASE Ligands: MR9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: MR9
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Crystal Structure Of Aminoquinazoline 1 Bound To Lck
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-02-27 Classification: TRANSFERASE Ligands: 242 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-02-27
Ligands: 242
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Crystal Structure Of Aminoquinazoline 36 Bound To Lck
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2007-02-27 Classification: TRANSFERASE Ligands: 1N8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-02-27
Ligands: 1N8
