Search Count: 19
![]() |
Human Mesotrypsin (Prss3) Unliganded And In An Active (E) Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2025-06-11 Classification: HYDROLASE Ligands: CA, CL, 2F2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-11
Ligands: CA, CL, 2F2
![]() |
Human Mesotrypsin (Prss3) Unliganded And In Autoinhibited (E*) Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-06-11 Classification: HYDROLASE Ligands: SO4, CA, ACT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-11
Ligands: SO4, CA, ACT, GOL
![]() |
Complex Of Tissue Inhibitor Of Metalloproteinases-1 (Timp-1) Mutant (L34G/M66S/E67Y/L133N/S155L) With Matrix Metalloproteinase-3 Catalytic Domain (Mmp-3Cd)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2022-03-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, ZN, CL, TRS, SO4, GOL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: CA, ZN, CL, TRS, SO4, GOL, ACT
![]() |
Complex Of Tissue Inhibitor Of Metalloproteinases-1 (Timp-1) Mutant (L34G/M66D/T98G/P131S/Q153N) With Matrix Metalloproteinase-3 Catalytic Domain (Mmp-3Cd)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2022-03-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: CA, ZN
![]() |
Human Mesotrypsin (Prss3) Complexed With Tissue Factor Pathway Inhibitor Variant (Tfpi1-Kd1-K15R-I17C-I34C)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2019-02-06 Classification: HYDROLASE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: SO4
![]() |
Crystal Structure Of Mesotrypsin In Complex With Appi-M17C/I18F/F34C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-02-06 Classification: PROTEIN FIBRIL Ligands: EDO, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: EDO, CA
![]() |
Structure Of Human Mesotrypsin In Complex With Appi Variant T11V/M17R/I18F/F34V
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-09-12 Classification: PROTEIN BINDING Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: EDO
![]() |
Combinatorial Engineering Of Proteolytically Resistant Appi Variants That Selectively Inhibit Human Kallikrein 6 For Cancer Therapy
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-05-30 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
![]() |
Combinatorial Engineering Of Proteolytically Resistant Appi Variants That Selectively Inhibit Human Kallikrein 6 For Cancer Therapy
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-05-30 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
![]() |
Mesotrypsin In Complex With Cleaved Amyloid Precursor Like Protein 2 Inhibitor (Aplp2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2016-11-09 Classification: Hydrolase/Hydrolase inhibitor Ligands: CA, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: CA, SO4
![]() |
Human Mesotrypsin In Complex With Amyloid Precursor Protein Inhibitor Variant Appi-M17G/I18F/F34V
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2016-05-04 Classification: Hyrdolase/Hydrolase inhibitor |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
![]() |
Human Cationic Trypsin G193R Mutant In Complex With Bovine Pancreatic Trypsin Inhibitor
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-07-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: SO4, CA |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2015-07-22
Ligands: SO4, CA
![]() |
Human Cationic Trypsin K97D Mutant In Complex With Bovine Pancreatic Trypsin Inhibitor (Bpti)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-07-22 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CA, SO4 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2015-07-22
Ligands: CA, SO4
![]() |
Human Mesotrypsin Complexed With Bikunin Kunitz Domain 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-10-15 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: CA
![]() |
Human Mesotrypsin Complexed With Hai-2 Kunitz Domain 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2014-10-15 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: NAG, CA
![]() |
Human Mesotrypsin Complexed With Bovine Pancreatic Trypsin Inhibitor Variant (Bpti-K15R/R17G)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: CA
![]() |
Human Mesotrypsin Complexed With Bovine Pancreatic Trypsin Inhibitor Variant (Bpti-K15R/R17D)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: CA
![]() |
Human Mesotrypsin Complexed With Bovine Pancreatic Trypsin Inhibitor(Bpti)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2007-12-11 Classification: hydrolase/hydrolase inhibitor Ligands: SO4 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: SO4
![]() |
Human Cationic Trypsin Complexed With Bovine Pancreatic Trypsin Inhibitor (Bpti)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2007-12-11 Classification: hydrolase/hydrolase inhibitor Ligands: CA, SO4 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: CA, SO4
