Search Count: 16
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Crystal Structure Of Bace1 In Complex With 2-Aminooxazoline 3-Aza-4-Fluoro-Xanthene Inhibitor 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-03-04 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, 3UT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-04
Ligands: IOD, GOL, 3UT
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Crystal Structure Of Bace1 In Complex With 2-Aminooxazoline 3-Azaxanthene Inhibitor 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-02-04 Classification: Hydrolase/hydrolase inhibitor Ligands: IOD, 43K, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: IOD, 43K, GOL
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Hydroxyethylamine-Based Inhibitors Of Bace1: P1-P3 Macrocyclization Can Improve Potency, Selectivity, And Cell Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2013-07-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1QT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-10
Ligands: 1QT
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Bace-1 Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2013-07-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1QU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-10
Ligands: 1QU
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Crystal Structure Of Bace1 In Complex With Hydroxyethylamine-Macrocyclic Inhibitor 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-07-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1R8, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-03
Ligands: 1R8, GOL, SO4
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Crystal Structure Of Bace1 In Complex With Hydroxyethylamine-Macrocyclic Inhibitor 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2013-07-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: IOD, 1R6, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-03
Ligands: IOD, 1R6, GOL
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Crystal Structure Of Bace1 In Complex With Hydroxyethylamine Inhibitor 37
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0K9, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 0K9, GOL
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Structure Of Bace-1 (Beta-Secretase) In Complex With (2R)-N-((2S,3R)-1-(Benzo[D][1,3]Dioxol-5-Yl)-3-Hydroxy-4-((S)-6'-Neopentyl-3',4'-Dihydrospiro[Cyclobutane-1,2'-Pyrano[2,3-B]Pyridine]-4'-Ylamino)Butan-2-Yl)-2-Methoxypropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-04-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: IOD, GOL, 0KN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-18
Ligands: IOD, GOL, 0KN
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Pde10A Crystal Structure Complexed With Novel Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2012-03-21 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, SO4, 0JQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: ZN, SO4, 0JQ
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Structure Of Bace-1 (Beta-Secretase) In Complex With (R)-3-(2-Amino-6-O-Tolylquinolin-3-Yl)-N-((R)-2,2-Dimethyltetrahydro-2H-Pyran-4-Yl)-2-Methylpropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, 3RS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, GOL, 3RS
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Structure Of Bace-1 (Beta-Secretase) In Complex With 6-(Thiophen-3-Yl)Quinolin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, RSV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, RSV
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Structure Of Bace-1 (Beta-Secretase) In Complex With 6-(2-(3,3-Dimethylbut-1-Ynyl)Phenyl)Quinolin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, RTH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, RTH
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Structure Of Bace-1 (Beta-Secretase) In Complex With 3-(2-Aminoquinolin-3-Yl)-N-Cyclohexyl-N-Methylpropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, RTM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, GOL, RTM
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Structure Of Bace-1 (Beta-Secretase) In Complex With 3-(2-Amino-6-O-Tolylquinolin-3-Yl)-N-Cyclohexylpropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, RTN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, GOL, RTN
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Structure Of Bace-1 (Beta-Secretase) In Complex With 3-(2-Aminoquinolin-3-Yl)-N-(Cyclohexylmethyl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, 3RU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, GOL, 3RU
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Structure Of Bace-1 (Beta-Secretase) In Complex With 2-((2-Amino-6-O-Tolylquinolin-3-Yl)Methyl)-N-(Cyclohexylmethyl)Pentanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, RVI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, GOL, RVI