Search Count: 19
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Il-1Beta In Complex With Macrocyclic Peptide Hit
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-05-22 Classification: CYTOKINE |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2024-05-22
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Il-1Beta In Complex With Covalent Del Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2024-05-22 Classification: CYTOKINE Ligands: A1H4A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-22
Ligands: A1H4A
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Human Il-1Beta, Unliganded
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2024-03-06 Classification: CYTOKINE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-06
Ligands: SO4
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X-Ray Structure Of Hdm2/Cmr19 At 1.45A: Discovery, X-Ray Structure And Cpp-Conjugation Enabled Uptake Of P53/Mdm2 Macrocyclic Peptide Inhibitors
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2021-09-22 Classification: LIGASE Ligands: SO4, CL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: SO4, CL
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 1: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HJW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HJW
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 2 At 2.3A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HKE, CHD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HKE, CHD
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 4 At 2.2A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HKZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HKZ
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 9 At 2.3A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HL8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HL8
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Rorgt (264-518;C455S) In Complex With The Fragment ("Cpd-1") And Rip140 Peptide At 1.80A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EE8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EE8
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Rorgt (264-518;C455S) In Complex With Inverse Agonist "Cpd-2" And Rip140 Peptide At 1.90A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EF5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EF5
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Rorgt (264-518;C455S) In Complex With Inverse Agonist "Cpd-9" And Rip140 Peptide At 1.66A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EEZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EEZ
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: C3S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: C3S
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-06-21 Classification: NUCLEAR PROTEIN Ligands: 99N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 99N
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: 98H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 98H
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: 98E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 98E
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: 444 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 444
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: 98N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 98N
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: 8YB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 8YB
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Synthesis And Biological Evaluation Of New Triazolo And Imidazolopyridine Rorgt Inverse Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2016-12-14 Classification: TRANSCRIPTION Ligands: Q6Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: Q6Y