Search Count: 9
 |
Discovery Of Bms-986144, A Third Generation, Pan Genotype Ns3/4A Protease Inhibitor For The Treatment Of Hepatitis C Virus Infection
Organism: Hepacivirus c
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-12-16 Classification: VIRAL PROTEIN Ligands: ZN, GXO |
Organism: Hepacivirus c
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: ZN, GXO
 |
Wdr5 In Complex With A Win Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-03-13 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HH7, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HH7, DMS, SO4
 |
Wdr5 In Complex With A Win Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2019-03-13 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HHM, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HHM, SO4, DMS
 |
Discovery Of Potent 2-Aryl-6,7-Dihydro-5Hpyrrolo[ 1,2-A]Imidazoles As Wdr5 Win-Site Inhibitors Using Fragment-Based Methods And Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLM
 |
Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLP
 |
Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLS, SO4
 |
Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLJ, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLJ, EPE
 |
Human Sterol 14-Alpha Demethylase (Cyp51) In Complex With Vfv In P1 Space Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-06-15 Classification: OXIDOREDUCTASE Ligands: HEM, VFV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-15
Ligands: HEM, VFV
 |
Human Sterol 14-Alpha Demethylase (Cyp51) In Complex With Vfv In C121 Space Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2016-06-08 Classification: OXIDOREDUCTASE Ligands: HEM, VFV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: HEM, VFV