Search Count: 18
![]() |
Cytochrome C Peroxidase Yhja
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2025-07-30 Classification: OXIDOREDUCTASE Ligands: HEC, HEM, CA, CL, EPE, SO4 |
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION
Release Date: 2025-07-30
Ligands: HEC, HEM, CA, CL, EPE, SO4
![]() |
Human Immunoproteasome 20S Particle In Complex With [2-(3-Ethylphenyl)-1-[(2S)-3-Phenyl-2-[(Pyrazin-2-Yl)Formamido]Propanamido]Ethyl]Boronic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2021-12-01 Classification: IMMUNE SYSTEM Ligands: SO4, NA, SKN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-01
Ligands: SO4, NA, SKN
![]() |
Crystal Structure Of Usp7 In Complex With A 4-Hydroxypiperidine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2018-04-11 Classification: HYDROLASE Ligands: SO4, GOL, CQ5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-11
Ligands: SO4, GOL, CQ5
![]() |
The Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-05-22 Classification: TRANSFERASE Ligands: C5I, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: C5I, EDO
![]() |
Jak2 Kinase (Jh1 Domain) In Complex With The Inhibitor Trans-4-[(8As)-2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(8Ah)-Yl]Cyclohexanecarbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J5
![]() |
Jak1 Kinase (Jh1 Domain) In Complex With The Inhibitor Trans-4-{2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(6H)-Yl}Cyclohexanecarbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J5
![]() |
Jak1 Kinase (Jh1 Domain) In Complex With The Inhibitor (Trans-4-{2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(6H)-Yl}Cyclohexyl)Acetonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J6
![]() |
Jak1 Kinase (Jh1 Domain) In Complex With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 15T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 15T
![]() |
The Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2012-07-04 Classification: Transferase/Transferase Inhibitor Ligands: JAK, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: JAK, EDO
![]() |
Jak1 Kinase (Jh1 Domain) In Complex With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2012-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: 0Q2
![]() |
Discovery And Optimization Of C-2 Methyl Imidazo-Pyrrolopyridines As Potent And Orally Bioavailable Jak1 Inhibitors With Selectivity Over Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2012-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1RS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: 1RS
![]() |
Discovery And Optimization Of C-2 Methyl Imidazo-Pyrrolopyridines As Potent And Orally Bioavailable Jak1 Inhibitors With Selectivity Over Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: JAK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: JAK
![]() |
Jak1 Kinase (Jh1 Domain) In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NH
![]() |
Jak2 Kinase (Jh1 Domain) In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NH
![]() |
Jak1 Kinase (Jh1 Domain) In Complex With Compound 49
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NL
![]() |
Jak1 Kinase (Jh1 Domain) In Complex With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NT, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NT, PEG
![]() |
Jak2 Kinase (Jh1 Domain) Triple Mutant In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NU, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NU, GOL
![]() |
Jak2 Kinase (Jh1 Domain) Triple Mutant In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NV
