Search Count: 27
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Crystal Structure Of D1228V C-Met Bound By Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: GOL, EDO, FMT, W49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: GOL, EDO, FMT, W49
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Crystal Structure Of D1228V C-Met Bound By Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: W3R, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: W3R, CL
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Crystal Structure Of D1228V C-Met Bound By Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: W3W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: W3W
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Crystal Structure Of D1228V C-Met Bound By Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: IOD, W3N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: IOD, W3N
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Crystal Structure Of Wild-Type C-Met Bound By Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: W40 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: W40
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Crystal Structure Of D1228V C-Met Bound By Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: W40 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: W40
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Mertk Kinase Domain With Type 1.5 Inhibitor Containing A Di-Methyl Pyrazole Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VJZ, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VJZ, CL, DMS
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Mertk Kinase Domain With Type 1.5 Inhibitor Containing A Di-Methyl, Cyano Pyrazole Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VK2, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VK2, CL, DMS
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Mertk Kinase Domain With Type 1.5 Inhibitor Containing A Tri-Methyl Pyrazole Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VK5, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VK5, CL
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Mertk Kinase Domain In Complex With Nps-1034
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4K
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Mertk Kinase Domain In Complex With Quinazoline-Based Inhbitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4E, SO4
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Mertk Kinase Domain In Complex With A Bisaminopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4N
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Mertk Kinase Domain In Complex With Purine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4Q
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Mertk Kinase Domain In Complex With A Type 2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4T
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Mertk Kinase Domain With Type 1.5 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4W
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Mertk Kinase Domain With Type 1 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4Z
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Mertk Kinase Domain With Type 3 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S5E, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S5E, CL, EDO
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Crystal Structure Of Wild-Type Cmet Bound By Foretinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-08-14 Classification: TRANSFERASE Ligands: CL, 88Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: CL, 88Z
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Crystal Structure Of D1228V Cmet Bound By Foretinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2019-08-14 Classification: TRANSFERASE Ligands: 88Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: 88Z
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Crystal Structure Of D1228V Cmet Bound By Bms-777607
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2019-08-14 Classification: TRANSFERASE Ligands: 353, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: 353, GOL
