Search Count: 26
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Bruton'S Tyrosine Kinase In Complex With Covalent Inhibitor Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2024-06-26 Classification: TRANSFERASE/INHIBITOR Ligands: UEO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: UEO
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Bruton'S Tyrosine Kinase In Complex With Covalent Inhibitor Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-06-26 Classification: TRANSFERASE/INHIBITOR Ligands: V72 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: V72
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Bruton'S Tyrosine Kinase In Complex With Covalent Inhibitor Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-06-26 Classification: TRANSFERASE/INHIBITOR Ligands: V7I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: V7I
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Structure Of Human Monoacylglycerol Lipase Bound To A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-03-14 Classification: Hydrolase/Hydrolase Inhibitor Ligands: E3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: E3A
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Pde2 Catalytic Domain Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2017-06-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 19F, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 19F, ZN, MG
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Pde2 Catalytic Domain Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-06-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7XS, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7XS, ZN, MG
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Pde2 Catalytic Domain Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-06-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7XV, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7XV, ZN, MG
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Pde2 Catalytic Domain Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2017-06-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, MG, 7Y1, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: ZN, MG, 7Y1, CL
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Pde2 Catalytic Domain Complexed With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2017-06-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 7Y4, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7Y4, ZN, MG
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Aminomethyl-Derived Beta Secretase (Bace1) Inhibitors: Engaging Gly230 Without An Anilide Functionality
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2017-01-11 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: P6U, IOD, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: P6U, IOD, EDO
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Aminomethyl-Derived Beta Secretase (Bace1) Inhibitors: Engaging Gly230 Without An Anilide Functionality
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2017-01-11 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 74B, IOD, NA, GOL, DMS, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 74B, IOD, NA, GOL, DMS, CL
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Structure Of Cytochrome P450 2D6 (Cyp2D6) Bace1 Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2017-01-11 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: HEM, ZN, P6U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: HEM, ZN, P6U
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Structure Of Cytochrome P450 2D6 (Cyp2D6) Bace1 Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2017-01-11 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: HEM, ZN, P6M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: HEM, ZN, P6M
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Crystal Structure Of Human Bace-1 Bound To Compound 24B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2015-03-04 Classification: Hydrolase/hydrolase inhibitor Ligands: 3VO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-04
Ligands: 3VO
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Crystal Structure Of Human Bace-1 Bound To Compound 36
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-03-04 Classification: Hydrolase/hydrolase inhibitor Ligands: 3VP, IOD, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-04
Ligands: 3VP, IOD, DMS
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Crystal Structure Of Human Bace-1 Bound To Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2015-03-04 Classification: Hydrolase/Hydrolase inhibitor Ligands: 3WP, IOD, NA, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-04
Ligands: 3WP, IOD, NA, GOL, DMS
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Human Pde9 In Complex With Selective Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-05-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, 0WF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: ZN, MG, 0WF
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Human Pde9 In Complex With Selective Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2013-05-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, 0WL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: ZN, MG, 0WL
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Human Phosphodiesterase 9 In Complex With Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-02-27 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, MG, 7RG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-27
Ligands: ZN, MG, 7RG
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Structure Of Pde10-Inhibitor Complex
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-06-15 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: SO4, ZN, MG, PFK |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: SO4, ZN, MG, PFK
