Search Count: 26
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Crystal Structure Of The Bromodomain Of Human Transcription Activator Brg1 (Smarca4) In Complex With 2-(6-Amino-5-(Piperazin-1-Yl)Pyridazin-3-Yl)Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2020-10-07 Classification: GENE REGULATION Ligands: FX5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: FX5, EDO
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Crystal Structure Of The Fifth Bromodomain Of Human Protein Polybromo-1 In Complex With 2-(6-Amino-5-(Piperazin-1-Yl)Pyridazin-3-Yl)Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2020-10-07 Classification: GENE REGULATION Ligands: FX5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: FX5, EDO
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Crystal Structure Of The Fifth Bromodomain Of Human Protein Polybromo-1 In Complex With Tert-Butyl 4-[3-Amino-6-(2-Hydroxyphenyl)Pyridazin-4-Yl]Piperazine-1-Carboxylate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-10-07 Classification: GENE REGULATION Ligands: QP8, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: QP8, EDO
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Protein Polybromo-1 (Pb1 Bd2) Bound To Mw278
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2020-08-26 Classification: PROTEIN BINDING Ligands: QMT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: QMT, EDO
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Protein Polybromo-1 (Pb1 Bd2) Bound To Dp28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.14 Å Release Date: 2020-08-26 Classification: PROTEIN BINDING Ligands: QMW, ZN, EDO, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: QMW, ZN, EDO, CL, ACT
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Crystal Structure Of Mllt1 (Enl) Yeats Domain In Complexed With Piperazine-Urea Derivative 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-11-06 Classification: TRANSCRIPTION Ligands: M7W, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: M7W, EDO
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Crystal Structure Of Mllt1 (Enl) Yeats Domain In Complexed With Piperazine-Urea Derivative 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2019-11-06 Classification: TRANSCRIPTION Ligands: EDO, M7T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: EDO, M7T
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Crystal Structure Of Mllt1 (Enl) Yeats Domain In Complexed With Piperazine-Urea Derivative 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-11-06 Classification: TRANSCRIPTION Ligands: EDO, M7N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: EDO, M7N
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Crystal Structure Of Mllt1 (Enl) Yeats Domain In Complexed With Benzimidazole-Amide Derivative 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-11-06 Classification: TRANSCRIPTION Ligands: M8K, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: M8K, EDO
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Crystal Structure Of Mllt1 (Enl) Yeats Domain In Complexed With Benzimidazole-Amide Derivative 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2019-11-06 Classification: TRANSCRIPTION Ligands: M7Z, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: M7Z, EDO
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Crystal Structure Of Mllt1 (Enl) Yeats Domain In Complexed With Benzimidazole-Amide Derivative 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-11-06 Classification: TRANSCRIPTION Ligands: M82, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: M82, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor 16I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2019-03-06 Classification: GENE REGULATION Ligands: EDO, HG5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-06
Ligands: EDO, HG5
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor 16K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-03-06 Classification: GENE REGULATION Ligands: HG8, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-06
Ligands: HG8, EDO
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Crystal Structure Of Enl (Mllt1) In Complex With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-11-28 Classification: TRANSCRIPTION Ligands: EDO, GKT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: EDO, GKT
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Crystal Structure Of Enl (Mllt1) In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-11-28 Classification: TRANSCRIPTION Ligands: EDO, GKQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: EDO, GKQ
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Crystal Structure Of Enl (Mllt1) In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-11-28 Classification: TRANSCRIPTION Ligands: EDO, SO4, GKN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: EDO, SO4, GKN
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Crystal Structure Of Enl (Mllt1) In Complex With Acetyllysine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-11-28 Classification: TRANSCRIPTION Ligands: EDO, ALY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: EDO, ALY
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Crystal Structure Of Enl (Mllt1), Apo Form
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2018-11-28 Classification: TRANSCRIPTION Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-28
Ligands: EDO
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Crystal Structure Of Mllt1 (Enl) Yeats Domain In Complexed With Compound 94
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-10-17 Classification: TRANSCRIPTION Ligands: SO4, EDO, GQ8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: SO4, EDO, GQ8
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Crystal Structure Of Mllt1 (Enl) Yeats Domain In Complexed With Sgc-Imllt (Compound 92)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-10-17 Classification: TRANSCRIPTION Ligands: SO4, EDO, GQ5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: SO4, EDO, GQ5
