Search Count: 29
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With Palazestrant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-03-19 Classification: TRANSCRIPTION Ligands: A1AEA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-19
Ligands: A1AEA, GOL
 |
Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3735967A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, I67, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: ZN, I67, EDO, GOL
 |
Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3543105A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAH, ZN, EDO, GOL, IO5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: SAH, ZN, EDO, GOL, IO5
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830334A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EDO, ZN, GOL, 96I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: EDO, ZN, GOL, 96I
 |
Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3852279B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, EDO, GOL, C79 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: ZN, EDO, GOL, C79
 |
Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Cofactor Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SAM, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: ZN, SAM, GOL, EDO
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAH, LUP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAH, LUP
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, EDO, SAM, L0J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, EDO, SAM, L0J
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, SAM, O41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, SAM, O41
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAM, O6A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAM, O6A
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Crystal Structure Of Human Phosphorylated Ire1Alpha In Complex With A Type Iii Kinase Inhibitor (Gsk2850163A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2015-11-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4K7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: 4K7
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Crystal Structure Of Pire1Alpha In Complex With Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2015-11-11 Classification: Transferase/transferase inhibitor Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: STU
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Crystal Structure Of Human Phosphorylated Ire1Alpha In Complex With Adp-Mg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2015-11-11 Classification: TRANSFERASE Ligands: MG, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: MG, ADP
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Crystal Structure Of Gsk6157 Bound To Perk (R587-R1092, Delete A660-T867) At 2.34A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2014-09-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 27D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 27D
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Crystal Structure Of Gsk6414 Bound To Perk (R587-R1092, Delete A660-T867) At 2.28 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 0WH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: GOL, 0WH
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Crystal Structure Of Gsk6924 Bound To Perk (R587-R1092, Delete A660-T867) At 2.70 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 924 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: 924
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Lead Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-06-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, JMZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-22
Ligands: GOL, SO4, JMZ
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Fragment8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: GOL, JNZ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: GOL, JNZ, SO4
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Fragment11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: GOL, SO4, JOZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: GOL, SO4, JOZ
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Phosphoinositide-Dependent Kinase-1 (Pdk1) With Fragment17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: GOL, SO4, JPZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: GOL, SO4, JPZ