Search Count: 8
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Pqr530 [(S)-4-(Difluoromethyl)-5-(4-(3-Methylmorpholino)-6-Morpholino-1,3,5-Triazin-2-Yl)Pyridin-2-Amine] Bound To The Pi3Ka Catalytic Subunit P110Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2019-06-26 Classification: TRANSFERASE Ligands: M1J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: M1J
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Pqr309 - A Potent, Brain-Penetrant, Orally Bioavailable, Pan-Class I Pi3K/Mtor Inhibitor As Clinical Candidate In Oncology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-09-06 Classification: TRANSFERASE Ligands: A3W, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-06
Ligands: A3W, SO4
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Orally Active Aminopyridines As Inhibitors Of Tetrameric Fructose 1,6- Bisphosphatase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-05-18 Classification: HYDROLASE Ligands: YCU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: YCU
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Orally Active Aminopyridines As Inhibitors Of Tetrameric Fructose 1,6- Bisphosphatase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-05-18 Classification: HYDROLASE Ligands: RO8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: RO8
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Fructose-1,6-Bisphosphatase(D-Fructose-1,6-Bisphosphate-1- Phosphohydrolase) (E.C.3.1.3.11) Complexed With An Amp Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2009-12-22 Classification: HYDROLASE Ligands: RO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-22
Ligands: RO3
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Fructose-1,6-Bisphosphatase(D-Fructose-1,6-Bisphosphate-1- Phosphohydrolase) (E.C.3.1.3.11) Complexed With An Amp Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-12-22 Classification: HYDROLASE Ligands: RO5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-22
Ligands: RO5
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Fructose-1,6-Bisphosphatase(D-Fructose-1,6-Bisphosphate -1- Phosphohydrolase) (E.C.3.1.3.11) Complexed With A Dual Binding Amp Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-07-22 Classification: HYDROLASE Ligands: R15 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-22
Ligands: R15
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Fructose-1,6-Bisphosphatase(D-Fructose-1,6-Bisphosphate -1- Phosphohydrolase) (E.C.3.1.3.11) Complexed With A Dual Binding Amp Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-07-22 Classification: HYDROLASE Ligands: ROK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-22
Ligands: ROK
