Search Count: 49
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Crystal Structure Of Human Exonuclease 1 (Exo1) With Dna And Compound 20
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-12-17 Classification: HYDROLASE Ligands: MG, NA, A1JNC, FMT |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-12-17
Ligands: MG, NA, A1JNC, FMT
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Crystal Structure Of Human Exonuclease 1 (Exo1) With Dna And Compound Art5537
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-12-17 Classification: HYDROLASE Ligands: MG, A1JO0, NA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-12-17
Ligands: MG, A1JO0, NA
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Structure Of Human Neutrophil Elastase In Complex With A 5,8-Dihydro[1,2,4]Triazolo[4,3-A]Pyrimidin-3(2H)-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.14 Å Release Date: 2025-12-10 Classification: HYDROLASE Ligands: NAG, FUC, A1JN2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-10
Ligands: NAG, FUC, A1JN2
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Crystal Structure Of Flap Endonuclease Fen1 With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2025-09-24 Classification: HYDROLASE Ligands: MG, EDO, A1JD4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-24
Ligands: MG, EDO, A1JD4
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Crystal Structure Of Flap Endonuclease Fen1 With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2025-09-24 Classification: HYDROLASE Ligands: A1JED, TEW, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-24
Ligands: A1JED, TEW, MG
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Crystal Structure Of Pi3K-Alpha In Complex With Taselisib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: 799 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: 799
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3W
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3R
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3N
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Crystal Structure Of Ternary Complex Of Pol Theta Polymerase Domain
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3
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Crystal Structure Of Pol Theta Polymerase Domain In Complex With Compound 5
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3, K7X |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3, K7X
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Crystal Structure Of Pol Theta Polymerase Domain In Complex With Compound 22
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: MG, DG3, K8I |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: MG, DG3, K8I
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Pi3K-Gamma K802T In Complex With Cpd 8 10-((1-(Tert-Butyl)Piperidin-4-Yl)Sulfinyl)-2-(1-Isopropyl-1H-1,2,4-Triazol-5-Yl)-5,6-Dihydrobenzo[F]Imidazo[1,2-D][1,4]Oxazepine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2017-11-15 Classification: TRANSFERASE/TRANSFERASE INHBITOR Ligands: BWY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-15
Ligands: BWY
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Egfr Kinase Domain Mutant "Tmlr" With Azabenzimidazole Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60B
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Egfr Kinase Domain Mutant "Tmlr" With 3-Carboxamide Azaindole Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60D
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Egfr Kinase Domain Mutant "Tmlr" With 3-Azetidinyl Azaindazole Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60E
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P110Alpha/P85Alpha With Compound 5
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-01-27 Classification: Transferase/Transferase Inhibitor Ligands: 5H2 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H2
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P110Alpha With Gdc-0326
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2016-01-27 Classification: Transferase/Inhibitor Ligands: 5H5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H5, EDO
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P110Delta/P85Alpha With Gdc-0326
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2016-01-27 Classification: Transferase/Inhibitor Ligands: 5H5 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H5
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Egfr Kinase Domain Mutant "Tmlr" With Pyridone Compound 2: 4-[2-(4-Chlorophenyl)Ethylamino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: 5Q2
