Search Count: 24
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Cdk2-Cycline1 In Complex With Allosteric Inhibitor I-198.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2024-01-31 Classification: CELL CYCLE/TRANSFERASE/INHIBITOR Ligands: A1AC4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
Ligands: A1AC4
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Cdk2-Cycline1 In Complex With Allosteric Inhibitor I-125A.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-01-31 Classification: CELL CYCLE/TRANSFERASE/INHIBITOR Ligands: A1AC5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
Ligands: A1AC5
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Crystal Structure Of Jak2 With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWP
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Crystal Structure Of Tyk2 With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWP
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Crystal Structure Of Tyk2 With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWM
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Structure Of Ciap With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2020-11-18 Classification: LIGASE Ligands: ZN, TKY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: ZN, TKY
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Ternary Complex Structure - Btk Ciap Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2020-11-18 Classification: LIGASE/TRANSFERASE Ligands: TL7, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: TL7, ZN
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Ternary Complex Structure - Btk Ciap Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.80 Å Release Date: 2020-11-18 Classification: LIGASE/TRANSFERASE Ligands: TKY, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: TKY, ZN
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Tyk2 With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: G5D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: G5D
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Tyk2 With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: G4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: G4J
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Jak1 With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: G4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: G4J
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Crystal Structure Of Egfr Kinase Domain (L858R, T790M, V948R) In Complex With The Covalent Inhibitor Co-1686
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.06 Å Release Date: 2017-10-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8OV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: 8OV
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Jak3 With Covalent Inhibitor 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KU
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Jak3 With Covalent Inhibitor 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KV, SO4
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Jak3 With Covalent Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2017-02-22 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7KX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 7KX
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Jak3 With Covalent Inhibitor Pf-06651600
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-11-09 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7H4, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 7H4, SO4
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Crystal Structure Of Mst3 With A Pyrrolopyrimidine Inhibitor (Pf-06447475)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2015-03-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MN, 3FE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: MN, 3FE
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Crystal Structure Of Mst3 With A Pyrrolopyrimidine Inhibitor (Pf-06454589).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2015-03-18 Classification: transferase/transferase inhibitor Ligands: 3JA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 3JA
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Structure Of Mst3 With A Pyrrolopyrimidine Inhibitor (Pf-06645342)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2015-03-18 Classification: transferase/transferase inhibitor Ligands: 3JB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 3JB
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Ck1D In Complex With 1-{4-[3-(4-Fluorophenyl)-1-Methyl-1H-Pyrazol-4-Yl]Pyridin-2-Yl}-N-Methylmethanamine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2013-09-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1QN, SO4, 1QO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: 1QN, SO4, 1QO
