Search Count: 5
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Bace1 In Complex With 4-(Cyclohexylamino)-1-(3-Fluorophenyl)-8-(3-Isopropoxybenzyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QA
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Bace1 In Complex With 8-(3-((1-Aminopropan-2-Yl)Oxy)Benzyl)-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-08-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: 4QD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QD
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Bace1 In Complex With 8-Benzyl-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-7-Methyl-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QF
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Discovery Of Pyrrolidine-Based B-Secretase Inhibitors: Lead Advancement Through Conformational Design For Maintenance Of Ligand Binding Efficiency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-01-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 508, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-18
Ligands: 508, SO4, GOL
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Crystal Structure Of Bace1 Bound To Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-02-03 Classification: HYDROLASE Ligands: SO4, GOL, 5MS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-03
Ligands: SO4, GOL, 5MS
