Search Count: 18
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Crebbp Bromodomain In Complex With Cpd3 ((S)-1-(3-(6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9U7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9U7
 |
Crebbp Bromodomain In Complex With Cpd8 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2018-03-07 Classification: TRANSFERASE/INHIBITOR Ligands: 9UA, DMS, GOL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UA, DMS, GOL
 |
Crebbp Bromodomain In Complex With Cpd10 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9UD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UD
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Crebbp Bromodomain In Complex With Cpd17 (N,2,7-Trimethyl-2,3-Dihydro-4H-Benzo[B][1,4]Oxazine-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: SO4, 9UG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: SO4, 9UG
 |
Lactate Dehydrogenase A In Complex With A Trisubstituted Piperidine-2,4-Dione Inhibitor Gne-140
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-18 Classification: Oxidoreductase/Oxidoreductase Inhibitor Ligands: NAD, SO4, GN0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: NAD, SO4, GN0
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Crystal Structure Of The Cbp Bromodomain In Complex With Cpi098
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 986, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 986, EDO
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Crystal Structure Of The Cbp Bromodomain In Complex With Cpi703
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING Ligands: 58N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 58N
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Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Sorafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BAX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: BAX
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Egfr Kinase Domain Mutant "Tmlr" With A Pyrazolopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 63M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: 63M
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Egfr Kinase Domain Mutant "Tmlr" With A Imidazopyridinyl-Aminopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 63N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: SO4, 63N
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Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Az628
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B1E, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: B1E, PEG
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Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Dabrafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: P06
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Crystal Structure Of Mek1 Kinase Bound To Gdc0973
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2013-08-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, EUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: ANP, MG, EUI
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B-Raf Kinase Domain In Complex With An Aminothienopyrimidine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: RI8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: RI8
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B-Raf Kinase Domain In Complex With An Aminopyridimine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: RI9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: RI9
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Human B-Raf Kinase Domain In Complex With An Bromopyridine Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TV4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: TV4
 |
Human B-Raf Kinase Domain In Complex With A Methoxypyrazolopyridinyl Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2011-10-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B0R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-05
Ligands: B0R
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Crystal Structure Of C-Raf (Raf-1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:4.00 Å Release Date: 2010-09-15 Classification: TRANSFERASE Ligands: SM5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: SM5