Search Count: 33
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Crystal Structure Of Gsk6157 Bound To Perk (R587-R1092, Delete A660-T867) At 2.34A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2014-09-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 27D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 27D
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Structure Of Dpp2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-09-19 Classification: HYDROLASE Ligands: NAG, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-19
Ligands: NAG, ZN
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Crystal Structure Of Gsk6414 Bound To Perk (R587-R1092, Delete A660-T867) At 2.28 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 0WH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: GOL, 0WH
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Crystal Structure Of Gsk6924 Bound To Perk (R587-R1092, Delete A660-T867) At 2.70 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 924 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-08
Ligands: 924
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Kinase Domain Of Insulin Receptor Complexed With A Pyrrolo Pyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-05-26 Classification: SIGNALING PROTEIN, TRANSFERASE Ligands: 351 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-05-26
Ligands: 351
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Insulin Receptor Kinase Complexed With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-12-30 Classification: TRANSFERASE Ligands: GS3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-30
Ligands: GS3
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Jnk1 Complexed With A Bis-Anilino-Pyrrolopyrimidine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-12-30 Classification: TRANSFERASE Ligands: GS7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-30
Ligands: GS7
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Insulin Receptor Kinase Complexed With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2008-12-23 Classification: TRANSFERASE Ligands: GS2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-23
Ligands: GS2
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Cdk2/Cyclina Complexed With A Pyrazolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2008-10-21 Classification: Transferase/Cell Cycle Ligands: PO5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-21
Ligands: PO5
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Cdk2/Cyclina Complexed With A Pyrazolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2008-10-21 Classification: Transferase/Cell cycle Ligands: 5BP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-21
Ligands: 5BP
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Ligand Binding Domain Of The Glucocorticoid Receptor Complexed With Fluticazone Furoate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2008-06-24 Classification: TRANSCRIPTION Ligands: GW6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-24
Ligands: GW6
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Erbb4 Kinase Domain Complexed With A Thienopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-03-18 Classification: TRANSFERASE Ligands: GW7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-18
Ligands: GW7
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Cathepsin K Complexed With A Semicarbazone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-08-08 Classification: HYDROLASE Ligands: CT1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-08
Ligands: CT1
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Cathepsin K Complexed With A Semicarbazone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2006-08-08 Classification: HYDROLASE Ligands: SO4, CT2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-08
Ligands: SO4, CT2
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Cathepsin K Complexed With A Pyrrolidine Ketoamide-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2006-03-21 Classification: HYDROLASE Ligands: 4PR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-21
Ligands: 4PR
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Cathepsin K Complexed With A Cyanamide-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2005-07-19 Classification: HYDROLASE Ligands: T2M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-07-19
Ligands: T2M
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Cathepsin K Complexed With A Constrained Ketoamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2005-07-19 Classification: HYDROLASE Ligands: SO4, 3FC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-07-19
Ligands: SO4, 3FC
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Cathepsin K Complexed With A Cyanopyrrolidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2005-03-22 Classification: HYDROLASE Ligands: NBL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-22
Ligands: NBL
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Cathepsin K Complexed With A Ketoamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2004-09-21 Classification: HYDROLASE Ligands: SO4, FSP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: SO4, FSP
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Cathepsin K Complexed With Carbamate Derivatized Norleucine Aldehyde
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2004-06-22 Classification: HYDROLASE Ligands: SO4, MYE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-06-22
Ligands: SO4, MYE
