Search Count: 26
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 20)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, PEG, WB4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, PEG, WB4
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Human Cation-Independent Mannose 6-Phosphate/ Igf2 Receptor Domains 9-10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-08-19 Classification: SUGAR BINDING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
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Human Cation-Independent Mannose 6-Phosphate/ Igf2 Receptor Domain 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2020-08-19 Classification: SUGAR BINDING PROTEIN Ligands: CL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: CL, NA
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Human Cation-Independent Mannose 6-Phosphate/Igf2 Receptor Domains 7-11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.47 Å Release Date: 2020-08-19 Classification: SUGAR BINDING PROTEIN Ligands: SO4, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: SO4, NAG
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Co-Structure Of Btk Kinase Domain With L-005085737 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULV, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULV, 5WE
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Co-Structure Of Btk Kinase Domain With L-005191930 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULY, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULY, 5WE
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Co-Structure Of Btk Kinase Domain With L-005298385 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: UM4, EDO, BTB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: UM4, EDO, BTB
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Discovery Of Mk-8353: An Orally Bioavailable Dual Mechanism Erk Inhibitor For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, G67 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SO4, G67
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Discovery Of 3(S)-Thiomethyl Pyrrolidine Erk Inhibitors For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-05-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SO4, F8V |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: SO4, F8V
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X-Ray Crystallographic Structure Of A High Affinity Igf2 Antagonist (Domain11 Ab5 Rhh) Based On Human Igf2R Domain 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-05-18 Classification: TRANSPORT PROTEIN Ligands: GOL, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: GOL, EDO, SO4
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Btk-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2016-03-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 5WH, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-23
Ligands: 5WH, 5WE
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Btk Kinase Domain With Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-02-03 Classification: TRANSFERASE Ligands: 5WF, 5WE, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 5WF, 5WE, CL, EDO
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Nmr Solution Structure Ensemble Of 3-4D Mutant Domain 11 Igf2R In Complex With Igf2 (Domain 11 Structure Only)
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2014-10-15 Classification: ANTITUMOR PROTEIN |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2014-10-15
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Nmr Solution Structure Ensemble Of 3-4D Mutant Domain 11 Igf2R
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2014-10-15 Classification: ANTITUMOR PROTEIN |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2014-10-15
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Nmr Solution Structure Ensemble Of Domain 11 Of The Echidna M6P/Igf2R Receptor
Organism: Tachyglossus aculeatus
Method: SOLUTION NMR Release Date: 2012-11-07 Classification: TRANSPORT PROTEIN |
Organism: Tachyglossus aculeatus
Method: SOLUTION NMR
Release Date: 2012-11-07
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Chicken Igf2R Domain 11
Organism: Gallus gallus
Method: SOLUTION NMR Release Date: 2012-02-15 Classification: TRANSPORT PROTEIN |
Organism: Gallus gallus
Method: SOLUTION NMR
Release Date: 2012-02-15
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Complex Structure Of E4 Mutant Human Igf2R Domain 11 Bound To Igf-Ii
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2012-02-15 Classification: TRANSPORT PROTEIN |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2012-02-15
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Mutated Domain 11 Of The Cytoplasmic Region Of The Cation-Independent Mannose-6-Phosphate Receptor
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2012-02-15 Classification: TRANSPORT PROTEIN |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2012-02-15
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Solution Structure Of Opossum Domain 11
Organism: Monodelphis domestica
Method: SOLUTION NMR Release Date: 2012-02-15 Classification: SIGNALING PROTEIN |
Organism: Monodelphis domestica
Method: SOLUTION NMR
Release Date: 2012-02-15
