Search Count: 24
![]() |
Crystal Structure Of Human Clk1 Kinase In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-11-06 Classification: SIGNALING PROTEIN Ligands: SO4, XQX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: SO4, XQX
![]() |
Crystal Structure Of Human Acvr1 (Alk2) Kinase In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2024-11-06 Classification: SIGNALING PROTEIN Ligands: SO4, XQX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: SO4, XQX
![]() |
Clathrin Terminal Domain Complexed With Pitstop 2C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2024-06-26 Classification: ENDOCYTOSIS Ligands: DMS, PEG, EDO, GOL, ACT, A1ATR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: DMS, PEG, EDO, GOL, ACT, A1ATR
![]() |
Clathrin Terminal Domain Complexed With Pitstop 2D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2024-06-26 Classification: ENDOCYTOSIS Ligands: DMS, TRS, PEG, ACT, EDO, GOL, A1ATQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: DMS, TRS, PEG, ACT, EDO, GOL, A1ATQ
![]() |
Room-Temperature X-Ray Structure Of Sars-Cov-2 Main Protease (3Cl Mpro) In Complex With A Non-Covalent Inhibitor Mcule-5948770040
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-03-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: YD1 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: YD1
![]() |
Rip2 Kinase Catalytic Domain Complex With 2(4[(1,3Benzothiazol5Yl)Amino]6(2Methylpropane2Sulfonyl)Quinazolin7Yl)Oxy)Ethyl Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2019-07-17 Classification: TRANSFERASE Ligands: K9T, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: K9T, CA
![]() |
Rip2 Kinase Catalytic Domain Complex With 2({4[(1,3Benzothiazol5Yl)Amino]6(2Methylpropane2Sulfonyl)Quinazolin7Yl}Oxy)Ethan1Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2019-07-17 Classification: TRANSFERASE Ligands: KA2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: KA2
![]() |
Crystal Structure Of Human Hexokinase 2 With Cmpd 30, A 2-Amino-6-Benzenesulfonamide Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 604 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 604
![]() |
Crystal Structure Of Human Hexokinase 2 With Cmpd 27, A 2-Amido-6-Benzenesulfonamide Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.92 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 603 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 603
![]() |
Crystal Structure Of Human Hexokinase 2 With Cmpd 1, A C-2-Substituted Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 62C, BG6, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 62C, BG6, FLC
![]() |
Insulin Co-Crystallizes In The Presence Of It Beta-Cell Chaperone Sulfatide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2015-02-11 Classification: HORMONE Ligands: ZN, CL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: ZN, CL, NA
![]() |
A Transforming Mutation In The Pleckstrin Homology Domain Of Akt1 In Cancer (Akt1-Ph_E17K)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2007-07-17 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-07-17
![]() |
A Transforming Mutation In The Pleckstrin Homology Domain Of Akt1 In Cancer (Akt1-Ph_E17K)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2007-07-17 Classification: TRANSFERASE Ligands: 4IP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-07-17
Ligands: 4IP
![]() |
Crystal Structure Of Cathepsin K Complexed With 7-Methyl-Substituted Azepan-3-One Compound
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2007-01-30 Classification: HYDROLASE Ligands: ILI |
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION
Release Date: 2007-01-30
Ligands: ILI
![]() |
Crystal Structure Of The Cysteine Protease Human Cathepsin K In Complex With A Covalent Azepanone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2003-01-14 Classification: HYDROLASE Ligands: 750 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-01-14
Ligands: 750
![]() |
Crystal Structure Of The Cysteine Protease Human Cathepsin K In Complex With A Covalent Azepanone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2003-01-14 Classification: HYDROLASE Ligands: 2CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-01-14
Ligands: 2CA
![]() |
C-Terminal Dna-Binding Domain Of Hiv-1 Integrase, Nmr, 42 Structures
Organism: Human immunodeficiency virus type 1 bh10
Method: SOLUTION NMR Release Date: 1999-12-14 Classification: TRANSFERASE |
Organism: Human immunodeficiency virus type 1 bh10
Method: SOLUTION NMR
Release Date: 1999-12-14
![]() |
Crystal Structure Of Cysteine Protease Human Cathepsin K In Complex With A Covalent Peptidomimetic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1999-06-08 Classification: HYDROLASE Ligands: I10 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1999-06-08
Ligands: I10
![]() |
Solution Structure Of The Guanine Nucleotide Exchange Factor Domain From Human Elongation Factor-One Beta, Nmr, 20 Structures
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 1999-05-18 Classification: GUANINE NUCLEOTIDE EXCHANGE FACTOR |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 1999-05-18
![]() |
Crystal Structure Of The Cysteine Protease Human Cathepsin K In Complex With A Covalent Pyrrolidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1998-10-14 Classification: HYDROLASE Ligands: PCM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1998-10-14
Ligands: PCM
