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Search Count: 15

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8EKX image
Structure Of Mbp-Mcl-1 In Complex With Mik665
Organism: Escherichia coli k-12, Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.55 Å Release Date: 2023-11-08
Classification: APOPTOSIS
Ligands: OK5

8EL1 image
Structure Of Mbp-Mcl-1 In Complex With Abbv-467
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.41 Å Release Date: 2023-10-25
Classification: APOPTOSIS
Ligands: WME

8EL0 image
Structure Of Mbp-Mcl-1 In Complex With A Macrocyclic Compound
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.92 Å Release Date: 2023-10-04
Classification: APOPTOSIS
Ligands: WLW

6VWC image
Crystal Structure Of Bcl-Xl In Complex With Tetrahydroisoquinoline-Pyridine Based Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.60 Å Release Date: 2020-10-21
Classification: APOPTOSIS/APOPTOSIS INHIBITOR
Ligands: RQ7

5KJ2 image
The Novel P300/Cbp Inhibitor A-485 Uncovers A Unique Mechanism Of Action To Target Ar In Castrate Resistant Prostate Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2017-09-27
Classification: transferase/transferase INHIBITOR
Ligands: 6TF, NA

5U2M image
Crystal Structure Of Human Nampt With A-1293201
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.89 Å Release Date: 2017-06-28
Classification: Transferase/Transferase Inhibitor
Ligands: 7T7, SO4

5U2N image
Crystal Structure Of Human Nampt With A-1326133
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.73 Å Release Date: 2017-06-28
Classification: Transferase/Transferase Inhibitor
Ligands: SO4, 7TA

5UF0 image
Brd4_Bd2-A-35165
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.35 Å Release Date: 2017-06-28
Classification: SIGNALING PROTEIN/INHIBITOR
Ligands: 89J

5UPE image
Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.93 Å Release Date: 2017-06-28
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 8HY

5UPF image
Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.69 Å Release Date: 2017-06-28
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 8HV

5UEU image
Brd4_Bd2_A-1107604
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.26 Å Release Date: 2017-05-10
Classification: SIGNALING PROTEIN/INHIBITOR
Ligands: 0S6

5UEW image
Brd2 Bromodomain2 With A-1360579
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.83 Å Release Date: 2017-05-10
Classification: SIGNALING PROTEIN/INHIBITOR
Ligands: 87D

5UEX image
Brd4_Bd2_A-1497627
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.29 Å Release Date: 2017-05-10
Classification: SIGNALING PROTEIN/INHIBITOR
Ligands: 89D

5UEY image
Brd4_Bd2_A-1412838
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.41 Å Release Date: 2017-05-10
Classification: SIGNALING PROTEIN/INHIBITOR
Ligands: 88M

5UEZ image
Brd4_Bd2_A-1342843
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.51 Å Release Date: 2017-05-10
Classification: SIGNALING PROTEIN/INHIBITOR
Ligands: 89G
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