Search Count: 23
![]() |
Pi3 Kinase Delta In Complex With 5-[3,6-Dihydro-2H-Pyran-4-Yl]-2-Methoxy-N-[2-Methylpyridin-4-Yl]Pyridine-3-Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7VT |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7VT
![]() |
Pi3 Kinase Delta In Complex With N-[2-(2-Fluoro-4-{[4-(Propan-2-Yl)Piperazin-1-Yl]Methyl}Phenyl)Pyridin-4-Yl]-2-Methoxy-5-(Morpholin-4-Yl)Pyridine-3-Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7XH |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7XH
![]() |
Pi3 Kinase Delta In Complex With 5-(3,6-Dihydro-2H-Pyran-4-Yl)-2-Methoxy-N-(5-{3-[4-(Propan-2-Yl)Piperazin-1-Yl]Prop-1-Yn-1-Yl}Pyridin-3-Yl)Pyridine-3-Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7XN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7XN
![]() |
Pi3 Kinase Delta In Complex With N-[5-(3,6-Dihydro-2H-Pyran-4-Yl)-2-Methoxypyridin-3-Yl]Benzenesulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2021-09-29 Classification: SIGNALING PROTEIN Ligands: 7XW |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: 7XW
![]() |
Pi3K Delta In Complex With N[5(7{2[4(2Hydroxypropan2Yl)Piperidin1 Yl]Ethoxy}1,3Dihydro2Benzofuran5Yl)2 Methoxypyridin3Yl]Methanesulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-01-01 Classification: TRANSFERASE Ligands: NQ2 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NQ2
![]() |
Pi3K Delta In Complex With 2Methoxyn[2Methoxy5(7{[(2R)4(Oxetan3 Yl)Morpholin2Yl]Methoxy}1,3Dihydro2 Benzofuran5Yl)Pyridin3Yl]Ethane1 Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-01-01 Classification: TRANSFERASE Ligands: NQ5 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NQ5
![]() |
Crystal Structure Of The Acvr1 (Alk2) Kinase In Complex With The Compound M4K2009
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2019-10-16 Classification: SIGNALING PROTEIN Ligands: M2Z, SO4, EDO, NH4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-16
Ligands: M2Z, SO4, EDO, NH4, DMS
![]() |
Pi3K Delta In Complex With N(2Chloro5Phenylpyridin3Yl)Benzenesulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2018-12-26 Classification: TRANSFERASE Ligands: HKQ |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: HKQ
![]() |
Pi3K Delta In Complex With N[2Chloro5(3,6Dihydro2Hpyran4Yl)Pyridin3Yl]Methanesulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2018-12-26 Classification: TRANSFERASE Ligands: HKK |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: HKK
![]() |
Pi3K Delta In Complex With 1Benzyln[5(3,6Dihydro2Hpyran4Yl)2Methoxypyridin3Yl]2Methyl1Himidazole4Sulfonamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2018-12-26 Classification: TRANSFERASE Ligands: HKN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: HKN
![]() |
Factor Xa Complex With Gtc000398
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-09-30 Classification: HYDROLASE Ligands: CA, 48W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: CA, 48W
![]() |
Factor Xa Complex With Gtc000401
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-09-30 Classification: HYDROLASE Ligands: CA, 4O1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: CA, 4O1
![]() |
Factor Xa Complex With Gtc000406
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-09-30 Classification: HYDROLASE Ligands: CA, MG, 4O6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: CA, MG, 4O6
![]() |
Factor Xa Complex With Gtc000422
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2015-09-30 Classification: HYDROLASE Ligands: CA, MG, 987 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: CA, MG, 987
![]() |
Factor Xa Complex With Gtc000441
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2015-09-30 Classification: HYDROLASE Ligands: CA, 44I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: CA, 44I
![]() |
Crystal Structure Of Mouse Pi3 Kinase Delta In Complex With Gsk2269557
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2015-09-16 Classification: TRANSFERASE Ligands: VVX |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: VVX
![]() |
Crystal Structure Of Mouse Pi3 Kinase Delta In Complex With Gsk2292767
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2015-09-16 Classification: TRANSFERASE Ligands: OKO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: OKO
![]() |
Catalytic Domain Of Human Phosphodiesterase 4B2B In Complex With A 5-Heterocycle Pyrazolopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2011-08-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, ARS, ZG1, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-03
Ligands: ZN, MG, ARS, ZG1, GOL
![]() |
Catalytic Domain Of Human Phosphodiesterase 4B2B In Complex With A 5-Heterocycle Pyrazolopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-08-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, ARS, ZG2, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-03
Ligands: ZN, MG, ARS, ZG2, GOL
![]() |
Crystal Structure Of Pde4B Catalytic Domain In Complex With A Pyrazolopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2009-05-19 Classification: HYDROLASE Ligands: ZN, MG, 20A, ARS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-05-19
Ligands: ZN, MG, 20A, ARS
