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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2026-03-04 Classification: TRANSLATION Ligands: MG, K, SPD, PUT, TRS, ZN |
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2026-03-04 Classification: TRANSLATION Ligands: K, PUT, SPD, A1B75, TRS, MG, ZN |
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Human 80S Ribosome Bound To Idb-002 Stalled On Fpak-Containing Nascent Chain
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2026-03-04 Classification: TRANSLATION Ligands: K, SPD, PUT, TRS, MG, A1B76, ZN |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-12-13 Classification: TRANSFERASE/INHIBITOR Ligands: O7I, SO4, EDO |
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Co-Structure Of Phosphatidylinositol 4,5-Bisphosphate 3-Kinase Catalytic Subunit Alpha Isoform And Brain Penetrant Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-07-19 Classification: TRANSFERASE Ligands: ZTV, SO4 |
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Co-Structure Phosphatidylinositol 4,5-Bisphosphate 3-Kinase Catalytic Subunit Alpha Isoform Complexed With Brain Penetrant Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2023-07-19 Classification: TRANSFERASE Ligands: ZUO |
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Structural Basis For Thalidomide Teratogenicity Revealed By The Cereblon-Ddb1-Sall4-Pomalidomide Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.58 Å Release Date: 2020-04-15 Classification: LIGASE Ligands: ZN, Y70 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2018-04-04 Classification: HORMONE RECEPTOR Ligands: C6V, GOL |
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Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2017-06-07 Classification: HYDROLASE Ligands: ZN, C90 |
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Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-06-07 Classification: HYDROLASE Ligands: ZN, 7TD, EPE |
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With (2E)-3-{4-[(1R)-2-(4-Fluorophenyl)-6-Hydroxy-1-Methy L-1,2,3,4- Tetrahydroisoquinolin-1-Yl]Phenyl}Prop-2-Enoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2017-03-29 Classification: HORMONE RECEPTOR Ligands: 77W |
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With (2E)-3-(4-{(1R)-6-Hydroxy-1-Methyl-2-[4-(Propan-2 -Yl)Phenyl]-1,2,3,4- Tetrahydroisoquinolin-1-Yl}Phenyl)Prop-2-Enoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2017-03-29 Classification: HORMONE RECEPTOR Ligands: 782 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-10-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 2UG |
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Crystal Structure Of Dipeptidyl-Peptidase 4 (Cd26, Adenosine Deaminase Complexing Protein 2) (Dpp-Iv-Wt) Complex With Bms-767778 Aka 2-(3-(Aminomethyl)-4-(2,4- Dichlorophenyl)-2-Methyl-5-Oxo-5,7-Dihydro-6H-Pyrrolo[3,4- B]Pyridin-6-Yl)-N,N-Dimethylacetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-09-04 Classification: HYDROLASE Ligands: 1MD |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2013-09-04 Classification: HYDROLASE Ligands: 1WH |
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Crystal Structure Of Human Dpp-Iv In Complex Withsa-(+)- Methyl2-(3-(Aminomethyl)-4-(2,4-Dichlorophenyl)-2-Methyl- 7-Oxo-5H-Pyrrolo[3,4-B]Pyridin-6(7H)-Yl)Acetate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-02-29 Classification: hydrolase/hydrolase inhibitor Ligands: NAG, LGE |
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Crystal Structure Of Human Dpp-Iv In Complex With Sa-(+)-3-(Aminomethyl)-4-(2,4-Dichlorophenyl)-6-(2-Methoxyphenyl)- 2-Methyl-5H-Pyrrolo[3,4-B]Pyridin-7(6H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-10-26 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, KXB |
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Crystal Structure Of Human Dpp-Iv In Complex With Sa-(+)-3-(Aminomethyl)-4-(2,4-Dichlorophenyl)-6-(2-Methoxyphenyl)- 2-Methyl-5H-Pyrrolo[3,4-B]Pyridin-7(6H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-10-26 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, KXA |
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Crystal Structure Of Human Dpp-Iv In Complex With Sa-(+)-(6-(Aminomethyl)-5-(2,4-Dichlorophenyl)-7-Methylimidazo[1,2-A]Pyrimidin-2-Yl)(Morpholino)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2010-08-11 Classification: HYDROLASE Ligands: NAG, 6A5, GOL |
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Crystal Structure Of The Rat Androgen Receptor Ligand Binding Domain Complex With An N-Aryl-Oxazolidin 2-Imine Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2009-04-28 Classification: HORMONE Ligands: LGB |




















