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9O3V image
Human 80S Ribosome Stalled On Myc Nascent Chain
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-03-04
Classification: TRANSLATION
Ligands: MG, K, SPD, PUT, TRS, ZN

9O3W image
Human 80S Ribosome Bound To Idb-001 Stalled On Myc Nascent Chain
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-03-04
Classification: TRANSLATION
Ligands: K, PUT, SPD, A1B75, TRS, MG, ZN

9O3Y image
Human 80S Ribosome Bound To Idb-002 Stalled On Fpak-Containing Nascent Chain
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-03-04
Classification: TRANSLATION
Ligands: K, SPD, PUT, TRS, MG, A1B76, ZN

8TUC image
Unphosphorylated Camkk2 In Complex With Cc-8977
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2023-12-13
Classification: TRANSFERASE/INHIBITOR
Ligands: O7I, SO4, EDO

8SBC image
Co-Structure Of Phosphatidylinositol 4,5-Bisphosphate 3-Kinase Catalytic Subunit Alpha Isoform And Brain Penetrant Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2023-07-19
Classification: TRANSFERASE
Ligands: ZTV, SO4

8SBJ image
Co-Structure Phosphatidylinositol 4,5-Bisphosphate 3-Kinase Catalytic Subunit Alpha Isoform Complexed With Brain Penetrant Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.10 Å Release Date: 2023-07-19
Classification: TRANSFERASE
Ligands: ZUO

6UML image
Structural Basis For Thalidomide Teratogenicity Revealed By The Cereblon-Ddb1-Sall4-Pomalidomide Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.58 Å Release Date: 2020-04-15
Classification: LIGASE
Ligands: ZN, Y70

6B0F image
Estrogen Receptor Alpha Ligand Binding Domain In Complex With Lsz102
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.86 Å Release Date: 2018-04-04
Classification: HORMONE RECEPTOR
Ligands: C6V, GOL

5U39 image
Pseudomonas Aeruginosa Lpxc In Complex With Chir-090

5U3B image
Pseudomonas Aeruginosa Lpxc In Complex With Nvs-Lpxc-01

5T92 image
Estrogen Receptor Alpha Ligand Binding Domain In Complex With (2E)-3-{4-[(1R)-2-(4-Fluorophenyl)-6-Hydroxy-1-Methy L-1,2,3,4- Tetrahydroisoquinolin-1-Yl]Phenyl}Prop-2-Enoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.22 Å Release Date: 2017-03-29
Classification: HORMONE RECEPTOR
Ligands: 77W

5T97 image
Estrogen Receptor Alpha Ligand Binding Domain In Complex With (2E)-3-(4-{(1R)-6-Hydroxy-1-Methyl-2-[4-(Propan-2 -Yl)Phenyl]-1,2,3,4- Tetrahydroisoquinolin-1-Yl}Phenyl)Prop-2-Enoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.00 Å Release Date: 2017-03-29
Classification: HORMONE RECEPTOR
Ligands: 782

4PH4 image
The Crystal Structure Of Human Vps34 In Complex With Pik-Iii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2014-10-29
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: GOL, 2UG

4JH0 image
Crystal Structure Of Dipeptidyl-Peptidase 4 (Cd26, Adenosine Deaminase Complexing Protein 2) (Dpp-Iv-Wt) Complex With Bms-767778 Aka 2-(3-(Aminomethyl)-4-(2,4- Dichlorophenyl)-2-Methyl-5-Oxo-5,7-Dihydro-6H-Pyrrolo[3,4- B]Pyridin-6-Yl)-N,N-Dimethylacetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2013-09-04
Classification: HYDROLASE
Ligands: 1MD

4LKO image
Crystal Structure Of Human Dpp-Iv In Complex With Bms-744891
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.43 Å Release Date: 2013-09-04
Classification: HYDROLASE
Ligands: 1WH

3Q0T image
Crystal Structure Of Human Dpp-Iv In Complex Withsa-(+)- Methyl2-(3-(Aminomethyl)-4-(2,4-Dichlorophenyl)-2-Methyl- 7-Oxo-5H-Pyrrolo[3,4-B]Pyridin-6(7H)-Yl)Acetate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2012-02-29
Classification: hydrolase/hydrolase inhibitor
Ligands: NAG, LGE

3SWW image
Crystal Structure Of Human Dpp-Iv In Complex With Sa-(+)-3-(Aminomethyl)-4-(2,4-Dichlorophenyl)-6-(2-Methoxyphenyl)- 2-Methyl-5H-Pyrrolo[3,4-B]Pyridin-7(6H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2011-10-26
Classification: HYDROLASE/HYDROLASE inhibitor
Ligands: NAG, KXB

3SX4 image
Crystal Structure Of Human Dpp-Iv In Complex With Sa-(+)-3-(Aminomethyl)-4-(2,4-Dichlorophenyl)-6-(2-Methoxyphenyl)- 2-Methyl-5H-Pyrrolo[3,4-B]Pyridin-7(6H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2011-10-26
Classification: HYDROLASE/HYDROLASE inhibitor
Ligands: NAG, KXA

3NOX image
Crystal Structure Of Human Dpp-Iv In Complex With Sa-(+)-(6-(Aminomethyl)-5-(2,4-Dichlorophenyl)-7-Methylimidazo[1,2-A]Pyrimidin-2-Yl)(Morpholino)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.34 Å Release Date: 2010-08-11
Classification: HYDROLASE
Ligands: NAG, 6A5, GOL

3G0W image
Crystal Structure Of The Rat Androgen Receptor Ligand Binding Domain Complex With An N-Aryl-Oxazolidin 2-Imine Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2009-04-28
Classification: HORMONE
Ligands: LGB
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