Search Count: 33
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Design And Synthesis Of P1-P3 Macrocyclic Tertiary Alcohol Comprising Hiv-1 Protease Inhibitors
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2013-11-06 Classification: HYDROLASE Ligands: CL, EQM |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: CL, EQM
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Design And Synthesis Of P1-P3 Macrocyclic Tertiary Alcohol Comprising Hiv-1 Protease Inhibitors
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2013-11-06 Classification: HYDROLASE Ligands: CL, M8Y |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: CL, M8Y
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Design And Synthesis Of P1-P3 Macrocyclic Tertiary Alcohol Comprising Hiv-1 Protease Inhibitors
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-11-06 Classification: HYDROLASE Ligands: CL, M8B |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: CL, M8B
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Potent Beta-Secretase 1 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-09-08 Classification: HYDROLASE Ligands: 929 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-08
Ligands: 929
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Potent Beta-Secretase 1 Hydroxyethylene Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-06-02 Classification: HYDROLASE Ligands: MV7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: MV7
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Crystal Structure Of Beta-Secretase 1 In Complex With Selective Beta-Secretase 1 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 586, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: 586, SO4
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Hiv-1 Protease Inhibitors Containing A Tertiary Alcohol In The Transition-State Mimic With Improved Cell-Based Antiviral Activity
Organism: Human immunodeficiency virus type 1 (z2/cdc-z34 isolate)
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2009-12-15 Classification: HYDROLASE Ligands: 5AH |
Organism: Human immunodeficiency virus type 1 (z2/cdc-z34 isolate)
Method: X-RAY DIFFRACTION
Release Date: 2009-12-15
Ligands: 5AH
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Hiv-1 Protease Inhibitors Containing A Tertiary Alcohol In The Transition-State Mimic With Improved Cell-Based Antiviral Activity
Organism: Human immunodeficiency virus type 1 (z2/cdc-z34 isolate)
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-12-15 Classification: HYDROLASE Ligands: 5AH |
Organism: Human immunodeficiency virus type 1 (z2/cdc-z34 isolate)
Method: X-RAY DIFFRACTION
Release Date: 2009-12-15
Ligands: 5AH
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Beta-Secretase 1 Complexed With Statine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-12-16 Classification: HYDROLASE Ligands: 757, IPA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-16
Ligands: 757, IPA
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Two-Carbon-Elongated Hiv-1 Protease Inhibitors With A Tertiary- Alcohol-Containing Transition-State Mimic
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2008-05-20 Classification: HYDROLASE Ligands: HI1 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2008-05-20
Ligands: HI1
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Two-Carbon-Elongated Hiv-1 Protease Inhibitors With A Tertiary- Alcohol-Containing Transition-State Mimic
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2008-05-20 Classification: HYDROLASE Ligands: HV1 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2008-05-20
Ligands: HV1
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P1' Extended Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol In The Transition-State Mimicking Scaffold
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-02-13 Classification: HYDROLASE Ligands: 1AH |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2007-02-13
Ligands: 1AH
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P1' Extended Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol In The Transition-State Mimicking Scaffold
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2007-02-13 Classification: HYDROLASE Ligands: 2AH |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2007-02-13
Ligands: 2AH
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P1' Extended Hiv-1 Protease Inhibitors Encompassing A Tertiary Alcohol In The Transition-State Mimicking Scaffold
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2007-02-13 Classification: HYDROLASE Ligands: 4AH |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2007-02-13
Ligands: 4AH
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Hiv-1 Protease In Complex With Inhibitor Aha455
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2005-12-14 Classification: HYDROLASE/INHIBITOR Ligands: A1A |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2005-12-14
Ligands: A1A
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Hiv-1 Protease In Complex With Fluoro Substituted Diol-Based C2- Symmetric Inhibitor
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2004-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: BE4 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2004-12-22
Ligands: BE4
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Hiv-1 Protease In Complex With Fluoro Substituted Diol-Based C2- Symmetric Inhibitor
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2004-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: BE5 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2004-12-22
Ligands: BE5
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Hiv-1 Protease In Complex With Fluoro Substituted Diol-Based C2- Symmetric Inhibitor
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2004-12-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: BE3 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2004-12-01
Ligands: BE3
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Hiv-1 Protease In Complex With Fluoro Substituted Diol-Based C2- Symmetric Inhibitor
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2004-10-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: BE6 |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2004-10-07
Ligands: BE6
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Hiv-1 Protease In Complex With The Inhibitor Bea435
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2002-06-26 Classification: HYDROLASE Ligands: BEH |
Organism: Human immunodeficiency virus
Method: X-RAY DIFFRACTION
Release Date: 2002-06-26
Ligands: BEH
