Search Count: 21
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Crystal Structure Of The Inha From Mycobacterium Tuberculosis In Complex With An12855, Ebsi 4333.
Organism: Mycobacterium tuberculosis (strain cdc 1551 / oshkosh)
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2018-05-16 Classification: OXIDOREDUCTASE Ligands: 9JA |
Organism: Mycobacterium tuberculosis (strain cdc 1551 / oshkosh)
Method: X-RAY DIFFRACTION
Release Date: 2018-05-16
Ligands: 9JA
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Crystal Structure Of The Inha From Mycobacterium Tuberculosis In Complex With An12855, Ebsi 4333.
Organism: Mycobacterium tuberculosis (strain cdc 1551 / oshkosh)
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2018-05-16 Classification: OXIDOREDUCTASE Ligands: 9JJ |
Organism: Mycobacterium tuberculosis (strain cdc 1551 / oshkosh)
Method: X-RAY DIFFRACTION
Release Date: 2018-05-16
Ligands: 9JJ
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Crystal Structure Of The Inha From Mycobacterium Tuberculosis In Complex With An12855, Ebsi 4333.
Organism: Mycobacterium tuberculosis (strain cdc 1551 / oshkosh)
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2018-05-16 Classification: OXIDOREDUCTASE Ligands: 9JM |
Organism: Mycobacterium tuberculosis (strain cdc 1551 / oshkosh)
Method: X-RAY DIFFRACTION
Release Date: 2018-05-16
Ligands: 9JM
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Chk1 Kinase Domain With Diazacarbazole Compound 8: N-[3-(6-Cyano-9H-Pyrrolo[2,3-B:5,4-C']Dipyridin-3-Yl)Phenyl]Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-06-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3XK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 3XK
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Chk1 Kinase Domain With Diazacarbazole Compound 7: 3-(2-Hydroxyphenyl)-9H-Pyrrolo[2,3-B:5,4-C']Dipyridine-6-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-06-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3XL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 3XL
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Chk1 Kinase Domain With Diazacarbazole Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2015-06-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3X7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 3X7
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Chk1 Kinase Domain In Complex With Diarylpyrazine Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2014-12-17 Classification: Transferase/Transferase Inhibitor Ligands: 3DL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: 3DL
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Chk1 Kinase Domain In Complex With Aminopyrazine Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2014-12-17 Classification: Transferase/Transferase Inhibitor Ligands: 3DV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: 3DV
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Chk1 Kinase Domain In Complex With Diazacarbazole Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2014-12-17 Classification: Transferase/Transferase Inhibitor Ligands: 3DW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: 3DW
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Chk1 Kinase Domain In Complex With Diazacarbazole Gne-783
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3DX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: 3DX
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Tyk2 (Jh1) In Complex With Adenosine Di-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2013-08-14 Classification: HYDROLASE Ligands: ADP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: ADP, MG
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Jak2 Kinase (Jh1 Domain) With 2,6-Dichloro-N-(2-Oxo-2,5-Dihydropyridin-4-Yl)Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-06-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0X2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: 0X2
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Tyk2 Kinase (Jh1 Domain) With 2,6-Dichloro-N-(2-Oxo-2,5-Dihydropyridin-4-Yl)Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-06-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, EDO, GOL, 0X2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: SO4, EDO, GOL, 0X2
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Tyk2 (Jh1) In Complex With 2,6-Dichloro-N-{2-[(Cyclopropylcarbonyl)Amino]Pyridin-4-Yl}Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-06-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0X5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: 0X5
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Jak2 Kinase (Jh1 Domain) In Complex With 2,6-Dichloro-N-{2-[(Cyclopropylcarbonyl)Amino]Pyridin-4-Yl}Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-06-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0X5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: 0X5
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Tyk2 (Jh1) In Complex With 2,6-Dichloro-4-Cyano-N-{2-[(Cyclopropylcarbonyl)Amino]Pyridin-4-Yl}Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2013-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0X6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 0X6
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Tyk2 (Jh1) In Complex With 2,6-Dichloro-N-[2-({[(1R,2R)-2-Fluorocyclopropyl]Carbonyl}Amino)Pyridin-4-Yl]Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0XH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 0XH
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Tyk2 (Jh1) In Complex With 2,6-Dichloro-4-Cyano-N-[2-({[(1R,2R)-2-Fluorocyclopropyl]Carbonyl}Amino)Pyridin-4-Yl]Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0XP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 0XP
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Crystal Structure Of Ciap1 Bir3 Bound To Gdc0152
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2012-02-22 Classification: Apoptosis Inhibitor Ligands: ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-22
Ligands: ZN
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Crystal Structure Of The Bir Domain Of Mliap Bound To Gdc0152
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2012-02-22 Classification: Apoptosis Inhibitor Ligands: ZN, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-22
Ligands: ZN, SO4
