Search Count: 37
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Structure Of Dcn1 Bound To N-((4S,5S)-3-(Aminomethyl)-7-Ethyl-4-(4-Fluorophenyl)-6-Oxo-1-Phenyl-4,5,6,7-Tetrahydro-1H-Pyrazolo[3,4-B]Pyridin-5-Yl)-3-(Trifluoromethyl)Benzamide
Organism: Enterobacteria phage rb59, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2021-07-14 Classification: LIGASE/Inhibitor Ligands: YHP |
Organism: Enterobacteria phage rb59, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: YHP
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Crystal Structure Of The Human Brd2 Bd1 Bromodomain In Complex With A Tetrahydroquinoline Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-11-13 Classification: Transcription/Inhibitor Ligands: G7V, SO4, EDO, 03S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-13
Ligands: G7V, SO4, EDO, 03S
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Crystal Structure Of The Human Brd2 Bd2 Bromodimain In Complex With A Tetrahydroquinoline Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2019-11-13 Classification: Transcription/Inhibitor Ligands: G7V, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-13
Ligands: G7V, EDO
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Structure Of Dcn1 Bound To N-((4S,5S)-7-Ethyl-4-(4-Fluorophenyl)-3-Methyl-6-Oxo-1-Phenyl-4,5,6,7-Tetrahydro-1H-Pyrazolo[3,4-B]Pyridin-5-Yl)-3-Methylbenzamide
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2019-09-11 Classification: LIGASE Ligands: MPD, O37 |
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-11
Ligands: MPD, O37
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Structure Of Dcn1 Bound To 3-Methyl-N-((4S,5S)-3-Methyl-6-Oxo-1-Phenyl-4-(P-Tolyl)-4,5,6,7-Tetrahydro-1H-Pyrazolo[3,4-B]Pyridin-5-Yl)Benzamide
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2019-09-11 Classification: LIGASE Ligands: O0A |
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-11
Ligands: O0A
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Structure Of (3S,4S)-1-Benzyl-4-(3-(3-(Trifluoromethyl)Phenyl)Ureido)Piperidin-3-Yl Acetate Bound To Dcn1
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2018-09-26 Classification: HYDROLASE, LIGASE/INHIBITOR Ligands: DOJ |
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: DOJ
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Structure Of 1-(Benzo[D][1,3]Dioxol-5-Ylmethyl)-1-(1-Propylpiperidin-4-Yl)-3-(3-(Trifluoromethyl)Phenyl)Urea Bound To Dcn1
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2018-09-26 Classification: HYDROLASE, LIGASE/INHIBITOR Ligands: DQD |
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: DQD
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Crystal Structure Of The Second Bromodomain Of Human Brd2 In Complex With A Tetrahydroquinoline Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2018-02-28 Classification: TRANSCRIPTION Ligands: SO4, EDO, 8J2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: SO4, EDO, 8J2
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With A Tetrahydroquinoline Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2018-02-28 Classification: TRANSCRIPTION Ligands: 8J2, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: 8J2, EDO
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Structure Of Dcn1 Bound To Nacm-Hit
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-05-24 Classification: LIGASE Ligands: 8Z7 |
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8Z7
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Structure Of Dcn1 Bound To Nacm-Opt
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2017-05-24 Classification: HYDROLASE Ligands: 8ZA |
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8ZA
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Structure Of Dcn1 Bound To Nacm-Cov
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2017-05-24 Classification: Ligase / protein binding Ligands: 8ZD |
Organism: Enterobacteria phage t4, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8ZD
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Structure Of Dcn4 Pony Domain Bound To Cul1 Whb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2017-05-24 Classification: Ligase / protein binding |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
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Targeting The Binding Function 3 Site Of The Androgen Receptor Through In Silico Molecular Modeling
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2011-12-07 Classification: TRANSCRIPTION Ligands: TES, SO4, 30Z |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: TES, SO4, 30Z
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Targeting The Binding Function 3 Site Of The Androgen Receptor Through In Silico Molecular Modeling
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-07-06 Classification: HORMONE RECEPTOR Ligands: TES, SO4, YLO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-07-06
Ligands: TES, SO4, YLO
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Targeting The Binding Function 3 Site Of The Androgen Receptor Through In Silico Molecular Modeling
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-07-06 Classification: HORMONE RECEPTOR Ligands: SO4, TES, 056 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-07-06
Ligands: SO4, TES, 056
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Targeting The Binding Function 3 Site Of The Androgen Receptor Through In Silico Molecular Modeling
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2011-07-06 Classification: HORMONE RECEPTOR Ligands: SO4, TES, YLQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-07-06
Ligands: SO4, TES, YLQ
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Thyroid Receptor Beta In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-02-26 Classification: HORMONE RECEPTOR Ligands: 4HY, LEG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-26
Ligands: 4HY, LEG, SO4
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Crystal Structure Of Ar Lbd With Shp Peptide Nr Box 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2007-12-04 Classification: TRANSCRIPTION Ligands: DHT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-04
Ligands: DHT
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Androgen Receptor Lbd With Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2007-09-25 Classification: HORMONE RECEPTOR Ligands: SO4, DHT, 2MI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, DHT, 2MI
