Search Count: 24
![]() |
Human Jnk2 Bound To Covalent Inhibitor Yl2056
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2023-06-28 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: Y56 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-28
Ligands: Y56
![]() |
Crystal Structure Of Amp-Bound Human Jnk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2022-06-22 Classification: TRANSFERASE Ligands: AMP, P6G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-22
Ligands: AMP, P6G
![]() |
Dgy-06-116, A Novel And Selective Covalent Inhibitor Of Src Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2019-07-31 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: HVY
![]() |
Crystal Structure Of Kras V14I-Gdp Demonstrating Open Switch 1 Conformation - Form 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-07-31 Classification: HYDROLASE Ligands: GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GDP
![]() |
Crystal Structure Of Kras V14I-Gdp Demonstrating Disorder Switch 1 Conformation - Form 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-07-31 Classification: HYDROLASE Ligands: GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GDP
![]() |
Src Kinase Bound To Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-02-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6H3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: 6H3
![]() |
Crystal Structure Of Erk2 Covalently Bound To Sm1-71
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: SO4, 6H3, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: SO4, 6H3, EDO, CL
![]() |
Crystal Structure Of Erk1 Covalently Bound To Sm1-71
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: 6H3, EWH, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: 6H3, EWH, SO4, EDO
![]() |
Crystal Structure Of Takinib Bound To Tak1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2017-08-30 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: EDH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-30
Ligands: EDH
![]() |
Crystal Structure Of Sm1-71 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2017-02-15 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6H3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: 6H3
![]() |
Crystal Structure Of Tl11-113 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-02-15 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6H4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: 6H4
![]() |
Crystal Structure Of Cpt1691 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2017-02-15 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6HF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: 6HF
![]() |
Crystal Structure Of Tl10-92 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2017-02-15 Classification: Transferase/Transferase Inhibitor Ligands: T92 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: T92
![]() |
Crystal Structure Of Tl11-128 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2017-02-15 Classification: Transferase/Transferase Inhibitor Ligands: 6L4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-15
Ligands: 6L4
![]() |
Glutathione S-Transferase Bound With Hydrolyzed Piperlongumine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2016-11-30 Classification: transferase/transferase inhibitor Ligands: 3LF, GSH, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: 3LF, GSH, MES
![]() |
Crystal Structure Of Tl10-81 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2016-09-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 5KW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 5KW
![]() |
Crystal Structure Of A Gdp-Bound G12R Oncogenic Mutant Of Human Gtpase Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.04 Å Release Date: 2015-06-10 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: GDP, MG
![]() |
Crystal Structure Of A Gdp-Bound G12V Oncogenic Mutant Of Human Gtpase Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2015-06-10 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: GDP, MG
![]() |
Crystal Structure Of A Gdp-Bound G13D Oncogenic Mutant Of Human Gtpase Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2015-06-10 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: GDP, MG
![]() |
Crystal Structure Of A Gdp-Bound Q61L Oncogenic Mutant Of Human Gt- Pase Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2015-06-10 Classification: signaling protein, hydrolase Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: GDP, MG
