Search Count: 21
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2025-10-01 Classification: TRANSFERASE Ligands: Y9T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-01
Ligands: Y9T
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2025-10-01 Classification: TRANSFERASE Ligands: A1JDR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-01
Ligands: A1JDR
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2025-10-01 Classification: TRANSFERASE Ligands: A1JDQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-01
Ligands: A1JDQ, SO4
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2022-05-04 Classification: TRANSFERASE Ligands: B8I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: B8I
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.03 Å Release Date: 2022-05-04 Classification: TRANSFERASE Ligands: B6I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: B6I
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2022-05-04 Classification: TRANSFERASE Ligands: B4U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: B4U
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-05-04 Classification: TRANSFERASE Ligands: B7R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: B7R
![]() |
Tricyclic Indazoles A Novel Class Of Selective Estrogen Receptor Degrader Antagonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2019-01-23 Classification: DNA BINDING PROTEIN Ligands: H8W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: H8W
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2018-05-23 Classification: SIGNALING PROTEIN Ligands: SO4, CJT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: SO4, CJT
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.67 Å Release Date: 2018-05-23 Classification: SIGNALING PROTEIN Ligands: SO4, CJQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: SO4, CJQ
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2018-05-23 Classification: SIGNALING PROTEIN Ligands: CJN, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: CJN, SO4
![]() |
Irak4 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2018-05-23 Classification: SIGNALING PROTEIN Ligands: CKN, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: CKN, SO4
![]() |
Irak4 In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2017-12-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 6QY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-06
Ligands: SO4, 6QY
![]() |
Irak4 In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2017-12-06 Classification: Transferase/Transferase Inhibitor Ligands: 6QX, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-06
Ligands: 6QX, SO4
![]() |
Irak4 In Complex With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2017-12-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6R1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-06
Ligands: 6R1
![]() |
Irak4 In Complex With Az3862
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-12-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 6R0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-06
Ligands: SO4, 6R0
![]() |
Irak4 In Complex With Az3864
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2017-12-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QZ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-06
Ligands: 6QZ, SO4
![]() |
11B-Hydroxysteroid Dehydrogenase Type I In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2014-09-03 Classification: OXIDOREDUCTASE Ligands: NAP, 4YQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: NAP, 4YQ
![]() |
11B-Hydroxysteroid Dehydrogenase Type I In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2014-03-05 Classification: OXIDOREDUCTASE Ligands: NAP, DZL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-05
Ligands: NAP, DZL
![]() |
Free-Wilson And Structural Approaches To Co-Optimising Human And Rodent Isoform Potency For 11B-Hydroxysteroid Dehydrogenase Type 1 11B-Hsd1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-11-28 Classification: OXIDOREDUCTASE Ligands: NAP, HD2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-28
Ligands: NAP, HD2
