Search Count: 20
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Crystal Structure Of Human Pi3Ka (P110A Subunit) With Mmv085400 Bound To The Active Site Determined At 2.9 Angstroms Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2022-05-04 Classification: TRANSFERASE/INHIBITOR Ligands: ZHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: ZHY
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Structure Of Sars Cov-2 Main Protease Shows Simultaneous Processing Of Its N- And C-Terminii
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2021-04-14 Classification: HYDROLASE |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
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Crystal Structure Of Pi3Kalpha Selective Inhibitor Pf-06843195
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VXY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VXY
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Crystal Structure Of Pi3Kalpha Selective Inhibitor 11-1575
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VY4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VY4
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Crystal Structure Of Pi3Kalpha Inhibitor 10-5429
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VY1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VY1
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Crystal Structure Of Pi3Kalpha Inhibitor 4-0686
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2021-01-06 Classification: SIGNALING PROTEIN, Transferase Ligands: VYP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-06
Ligands: VYP
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Structure Of The Axl Kinase Domain In Complex With A Macrocyclic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2017-07-26 Classification: Transferase/Transferase Inhibitor Ligands: 7YS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-26
Ligands: 7YS
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Crystal Structure Of The Mer Kinase Domain In Complex With A Macrocyclic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-07-26 Classification: Transferase/Transferase Inhibitor Ligands: 7YS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-26
Ligands: 7YS
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X-Ray Structure Of C-Met Kinase In Complex With Inhibitor 6-((6-(4- Fluorophenyl)-(1,2,4)Triazolo(4,3-B)(1,2,4)Triazin-3-Yl)Methyl) Quinoline.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-11-27 Classification: TRANSFERASE Ligands: 6XE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: 6XE
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X-Ray Structure Of C-Met Kinase In Complex With Inhibitor (S)-6-(1-(6- (1-Methyl-1H-Pyrazol-4-Yl)-(1,2,4)Triazolo(4,3-B)Pyridazin-3-Yl)Ethyl) Quinoline.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-11-27 Classification: TRANSFERASE Ligands: W9Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: W9Z
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X-Ray Structure Of C-Met Kinase In Complex With Inhibitor (S)-3-(1-(1H-Pyrrolo(2,3-B)Pyridin-3-Yl)Ethyl)-N-Isopropyl-(1,2,4)Triazolo(4,3- B)Pyridazin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2013-11-27 Classification: TRANSFERASE Ligands: 5TF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: 5TF
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Crystal Structure Of C-Met Kinase Domain In Complex With 4-(3-((1H- Pyrrolo(2,3-B)Pyridin-3-Yl)Methyl)-(1,2,4)Triazolo(4,3-B)(1,2,4) Triazin-6-Yl)Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-09-26 Classification: TRANSFERASE Ligands: 4K0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-26
Ligands: 4K0
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Crystal Structure Of C-Met Kinase Domain In Complex With 4-((6-(4- Fluorophenyl)-(1,2,4)Triazolo(4,3-B)(1,2,4)Triazin-3-Yl)Methyl)Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-09-26 Classification: TRANSFERASE Ligands: F47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-26
Ligands: F47
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Crystal Structure Of C-Met Kinase Domain In Complex With N'-((3Z)-4- Chloro-7-Methyl-2-Oxo-1,2-Dihydro-3H-Indol-3-Ylidene)-2-(4- Hydroxyphenyl)Propanohydrazide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2011-09-14 Classification: TRANSFERASE Ligands: 6XP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-14
Ligands: 6XP
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X-Ray Structure Of Pf-04217903 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-08-31 Classification: TRANSFERASE Ligands: KRW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: KRW
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Structure Of The Human Anaplastic Lymphoma Kinase In Complex With Crizotinib (Pf-02341066)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-09-15 Classification: TRANSFERASE Ligands: VGH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: VGH
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X-Ray Structure Of Pha-00665752 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-08-25 Classification: TRANSFERASE Ligands: PFY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-25
Ligands: PFY
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X-Ray Structure Of Pf-02341066 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-06-02 Classification: TRANSFERASE Ligands: VGH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-06-02
Ligands: VGH
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Structure Of Catalytic Domain Of Human Protein Kinase C Beta Ii Complexed With A Bisindolylmaleimide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2006-11-14 Classification: TRANSFERASE Ligands: PDS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-14
Ligands: PDS
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Crystal Structure Of Nadp-Dependent Isocitrate Dehydrogenase From Porcine Heart Mitochondria
Organism: Sus scrofa
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2002-11-13 Classification: OXIDOREDUCTASE Ligands: MN, ICT, SO4 |
Organism: Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2002-11-13
Ligands: MN, ICT, SO4
