Search Count: 9
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Human Glucokinase In Complex With Novel Indazole Activator.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2017-05-31 Classification: transferase/transferase activator Ligands: GLC, 8WM, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: GLC, 8WM, IOD
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Human Glucokinase In Complex With Novel Pyrazole Activator.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2017-05-31 Classification: transferase/transferase activator Ligands: GLC, 8WJ, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: GLC, 8WJ, IOD
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Coactivator-Associated Arginine Methyltransferase 1 With Tp-064
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-12-21 Classification: TRANSFERASE Ligands: SAH, 7VM, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: SAH, 7VM, UNX
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Discovery Of Tak-659, An Orally Available Investigational Inhibitor Of Spleen Tyrosine Kinase (Syk)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2016-11-30 Classification: Transferase/Transferase Inhibitor Ligands: 7KG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: 7KG, EDO
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Discovery Of Tak-659, An Orally Available Investigational Inhibitor Of Spleen Tyrosine Kinase (Syk)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2016-11-30 Classification: Transferase/Transferase Inhibitor Ligands: 7KF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: 7KF
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With Syr-472
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2016-07-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 6RL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-13
Ligands: NAG, 6RL
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Parp Complexed With Benzo[1,4]Oxazin-3-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-08-07 Classification: transferase/transferase inhibitor Ligands: 1WQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: 1WQ
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Crystal Structure Of Human Hdac2 Complexed With An N-(2-Aminophenyl)Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2010-04-28 Classification: HYDROLASE Ligands: ZN, CA, NA, LLX, NHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-28
Ligands: ZN, CA, NA, LLX, NHE
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Tyrosine-48 Is The Proton Donor And Histidine-110 Directs Substrate Stereochemical Selectivity In The Reduction Reaction Of Human Aldose Reductase: Enzyme Kinetics And The Crystal Structure Of The Y48H Mutant Enzyme
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 1994-07-31 Classification: OXIDOREDUCTASE Ligands: NAP, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1994-07-31
Ligands: NAP, CIT
