Search Count: 15
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Crystal Structure Of Trim33 Phd-Bromodomain Isoform B In Complex With H3K10Ac Histone Peptide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-06-29 Classification: TRANSCRIPTION Ligands: EDO, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-29
Ligands: EDO, ZN
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 10B.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FKY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: FKY
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 13B.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22L, GO7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: 22L, GO7
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 19.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 22L, GOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: 22L, GOD
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Crystal Structure Of Trk-A In Complex With The Pan-Trk Kinase Inhibitor, Compound 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2018-07-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GXA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-11
Ligands: GXA
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Crystal Structure Of Tyrosine-Protein Kinase Receptor In Complex With 2,4-Dichloro-N-(3-Methyl-1-Phenyl-1H-Pyrazol-5-Yl)Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2018-05-02 Classification: TRANSFERASE/Inhibitor Ligands: FQJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: FQJ
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Crystal Structure Of Tyrosine-Protein Kinase Receptor In Complex With 5-(4-Fluorophenyl)Thieno[2,3-D]Pyrimidin-4(3H)-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2018-05-02 Classification: TRANSFERASE/Inhibitor Ligands: FQD, GOL, FQM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: FQD, GOL, FQM
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Crystal Structure Of Tyrosine-Protein Kinase Receptor In Complex With 5-(4-Fluorophenyl)Thieno[2,3-D]Pyrimidin-4(3H)-One And 5-{[2,4-Dichloro-5-(Pyridin-2-Yl)Benzene-1-Carbonyl]Amino}-N-(2-Hydroxy-2-Methylpropyl)-1-Phenyl-1H-Pyrazole-3-Carboxamide Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2018-05-02 Classification: TRANSFERASE/Inhibitor Ligands: FQD, FQG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: FQD, FQG
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Crystal Structure Of Tyrosine-Protein Kinase Receptor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2018-05-02 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
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Kinase Domain Mutant Of Human Itk In Complex With A Covalently-Binding Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2013-08-21 Classification: Transferase/Transferase inhibitor Ligands: G5K, G6K, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-21
Ligands: G5K, G6K, SO4, GOL
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Setd7 In Complex With Inhibitor (R)-Pfi-2 And S-Adenosyl-Methionine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-04-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 1L8, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-17
Ligands: SAM, 1L8, UNX
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Crystal Structure Of The First Bromodomain Of Human Brd2 With The Inhibitor Gw841819X
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-06-15 Classification: NUCLEAR PROTEIN Ligands: WSH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: WSH, SO4
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Crystal Structure Of The First Bromodomain Of Human Brd2 With The Inhibitor Gsk525762 (Ibet)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2011-06-15 Classification: SIGNALING PROTEIN Ligands: EAM, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: EAM, SO4
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Crystal Structure Of The First Bromodomain Of Human Brd4 With The Inhibitor Gw841819X
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2011-06-15 Classification: SIGNALING PROTEIN Ligands: EDO, WSH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: EDO, WSH
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Crystal Structure Of The Second Bromodomain Of Human Brd4 With The Inhibitor Gw841819X
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-06-15 Classification: SIGNALING PROTEIN Ligands: WSH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: WSH
