Search Count: 21
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Discovery Of Novel 7-Azaindoles As Pdk1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: SO4, 61Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: SO4, 61Y
 |
Discovery Of Novel 7-Azaindoles As Pdk1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: SO4, 62O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: SO4, 62O
 |
Discovery Of Novel 7-Azaindoles As Pdk1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: 63L, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 63L, SO4
 |
Discovery Of Novel 7-Azaindoles As Pdk1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: 63E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 63E, SO4
 |
Selection Of Fragments For Kinase Inhibitor Design: Decoration Is Key
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2015-10-28 Classification: Transferase/Transferase Inhibitor Ligands: 3WJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 3WJ, SO4
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Selection Of Fragments For Kinase Inhibitor Design: Decoration Is Key
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2015-08-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3WK, SO4, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: 3WK, SO4, TRS
 |
Selection Of Fragments For Kinase Inhibitor Design: Decoration Is Key
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2014-12-24 Classification: TRANSFERASE Ligands: 3WA, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3WA, SO4
 |
Selection Of Fragments For Kinase Inhibitor Design: Decoration Is Key
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2014-12-24 Classification: TRANSFERASE Ligands: 3WN, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3WN, SO4
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Selection Of Fragments For Kinase Inhibitor Design: Decoration Is Key
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2014-12-24 Classification: TRANSFERASE Ligands: 3WO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3WO, SO4
 |
Selection Of Fragments For Kinase Inhibitor Design: Decoration Is Key
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-12-24 Classification: TRANSFERASE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: SO4
 |
Selection Of Fragments For Kinase Inhibitor Design: Decoration Is Key
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-12-24 Classification: TRANSFERASE Ligands: 3WR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3WR
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Fragment-Based Discovery Of Focal Adhesion Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2013-09-11 Classification: Transferase/Transferase Inhibitor Ligands: K8A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: K8A
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Focal Adhesion Kinase Catalytic Domain In Complex With 1-[4-(6-Amino-Purin-9-Yl)-Phenyl]-3-(5-Tert-Butyl-2-P-Tolyl-2H-Pyrazol-3-Yl)-Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-09-11 Classification: Transferase/Transferase Inhibitor Ligands: K9Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: K9Y
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Focal Adhesion Kinase Catalytic Domain In Complex With 3-Methyl-1,4-Dihydro-Pyrazolo[4,5-C]Pyrazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2013-09-11 Classification: Transferase/Transferase Inhibitor Ligands: 4KA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: 4KA
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Focal Adhesion Kinase Catalytic Domain In Complex With 1-(5-Tert-Butyl-2-P-Tolyl-2H-Pyrazol-3-Yl)-3-(4-Pyridin-3- Yl-Phenyl)-Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2013-09-11 Classification: Transferase/Transferase Inhibitor Ligands: KAO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: KAO, SO4
 |
Focal Adhesion Kinase Catalytic Domain In Complex With N-{3-[(5-Cyano-2-Phenyl-1H-Pyrrolo[2,3-B]Pyridin-4-Ylamino)- Methyl]-Pyridin-2-Yl}-N-Methyl-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2013-09-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 10N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-04
Ligands: 10N
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Focal Adhesion Kinase Catalytic Domain In Complex With (2-Fluoro-Phenyl)-(1H-Pyrazolo[3,4-D]Pyrimidin-4-Yl)-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-09-04 Classification: TRANSFERASE Ligands: 4GU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-04
Ligands: 4GU
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Structural And Biophysical Characterization Of The Syk Activation Switch
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2012-11-28 Classification: TRANSFERASE Ligands: ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-28
Ligands: ANP, MG
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Structural And Biophysical Characterization Of The Syk Activation Switch
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2012-11-28 Classification: TRANSFERASE Ligands: MG, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-28
Ligands: MG, ANP
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Structural And Biophysical Characterization Of The Syk Activation Switch
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-11-28 Classification: TRANSFERASE Ligands: ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-28
Ligands: ANP, MG