Search Count: 72
![]() |
Kat6A Myst Domain Complexed With A H3K14-Coa Bisubstrate Inhibitor
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2025-02-19 Classification: TRANSFERASE/INHIBITOR Ligands: CMC, ZN, GOL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: CMC, ZN, GOL
![]() |
Crystal Structure Of Mastl Kinase Domain In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2025-01-22 Classification: TRANSFERASE/INHIBITOR Ligands: A1AAE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: A1AAE
![]() |
Crystal Structure Of Map4K4 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2025-01-22 Classification: TRANSFERASE/INHIBITOR Ligands: A1AAA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: A1AAA
![]() |
Structure Of Sars-Cov-2 Mpro Mutant (S144A) In Complex With Nirmatrelvir (Pf-07321332)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2024-08-07 Classification: VIRAL PROTEIN, HYDROLASE/INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-08-07
Ligands: 4WI
![]() |
Structure Of Sars-Cov-2 Mpro Mutant (A173V) In Complex With Nirmatrelvir (Pf-07321332)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2024-08-07 Classification: VIRAL PROTEIN, HYDROLASE/INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-08-07
Ligands: 4WI
![]() |
Structure Of Sars-Cov-2 Mpro Mutant (A173V,T304I)) In Complex With Nirmatrelvir (Pf-07321332)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2024-08-07 Classification: VIRAL PROTEIN, HYDROLASE/INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-08-07
Ligands: 4WI
![]() |
Structure Of Sars-Cov-2 Mpro Mutant (T21I,S144A,T304I) In Complex With Nirmatrelvir (Pf-07321332)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2024-08-07 Classification: VIRAL PROTEIN, HYDROLASE/INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-08-07
Ligands: 4WI
![]() |
Structure Of Sars-Cov-2 Mpro Mutant (T21I,T304I)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2024-08-07 Classification: VIRAL PROTEIN, HYDROLASE |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-08-07
![]() |
Structure Of Sars-Cov-2 Mpro Mutant (L50F,T304I)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2024-08-07 Classification: VIRAL PROTEIN, HYDROLASE Ligands: HOH |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-08-07
Ligands: HOH
![]() |
Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-05-15 Classification: VIRAL PROTEIN Ligands: YDL |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-05-15
Ligands: YDL
![]() |
Crystal Structure Of Kat6A In Complex With Inhibitor Ctx-648 (Pf-9363)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2023-07-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R7L, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: R7L, ZN
![]() |
Structure Of Sars-Cov-2 Mpro Lambda (G15S) In Complex With Nirmatrelvir (Pf-07321332)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2022-03-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2022-03-09
Ligands: 4WI
![]() |
Structure Of Sars-Cov-2 Mpro Mutant (K90R) In Complex With Nirmatrelvir (Pf-07321332)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2022-03-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2022-03-09
Ligands: 4WI
![]() |
Structure Of Sars-Cov-2 Mpro Omicron P132H In Complex With Nirmatrelvir (Pf-07321332)
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-01-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: 4WI
![]() |
Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4W8 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4W8
![]() |
Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4WI
![]() |
Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4YG |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4YG
![]() |
Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2021-11-10 Classification: HYDROLASE/INHIBITOR Ligands: 4WI |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: 4WI
![]() |
Crystal Structure Of Human Naa50 In Complex With A Cofactor Derived Inhibitor (Compound 1)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: COA
![]() |
Crystal Structure Of Human Naa50 In Complex With A Truncated Cofactor Derived Inhibitor (Compound 2)
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: U44 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-07-01
Ligands: U44
