Search Count: 59
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Crystal Structure Of Human Wrn Helicase With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2026-05-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, A1C4J, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-13
Ligands: ZN, A1C4J, EDO
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Crystal Structure Of Human Wrn Helicase With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2026-05-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, A1C4L, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-13
Ligands: ZN, A1C4L, CL, EDO
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Crystal Structure Of Human Wrn Helicase With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2026-05-13 Classification: HYDROLASE Ligands: A1C4O, ATP, ZN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-13
Ligands: A1C4O, ATP, ZN, EDO
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Human P300 Complexed With A Proline-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EDO, C0C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ZN, EDO, C0C
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Human P300 Complexed With A Glycine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EDO, C3I, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ZN, EDO, C3I, ACT
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Human P300 Complexed With An Azaindazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ETL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ETL
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Tnni3K Complexed With N-Methyl-4-(4-(3-(3-(Trifluoromethyl) Phenyl) Ureido) Phenoxy)Picolinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2021-11-10 Classification: TRANSFERASE/INHIBITOR Ligands: ZFS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: ZFS
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Tnni3K Complexed With 1-(3,5-Dichloro-4-((6-(Methylamino)Pyrimidin-4-Yl)Oxy)Phenyl)-3-(3-(Trifluoromethyl)Phenyl)Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2021-11-10 Classification: TRANSFERASE/INHIBITOR Ligands: ZGD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: ZGD
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: SAH, ZN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: SAH, ZN, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, X52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, X52
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3685032A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, UXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, UXM
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAH, LUP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAH, LUP
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, EDO, SAM, L0J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, EDO, SAM, L0J
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, SAM, O41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, SAM, O41
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAM, O6A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAM, O6A
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Tnni3K Complexed With A 4,6-Diaminopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.97 Å Release Date: 2018-04-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CV4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: CV4
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Co-Crystal Structure Of Human Smyd3 With An Aza-Sah Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-03-30 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, MG, DMS, 62X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: ZN, MG, DMS, 62X
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Co-Crystal Structure Of Human Smyd3 With A Mekk2 Peptide At 2.13A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2016-03-30 Classification: TRANSFERASE Ligands: ZN, MG, EDO, SAH, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: ZN, MG, EDO, SAH, GOL
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Braf Complexed With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2016-03-16 Classification: Transferase/Transferase Inhibitor Ligands: GOL, 4EF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-16
Ligands: GOL, 4EF
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Tnni3K Complexed With Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.07 Å Release Date: 2015-09-23 Classification: Transferase/Transferase Inhibitor Ligands: 4CV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-23
Ligands: 4CV
