Search Count: 20
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Crystal Structure Of C-Met Mutant Y1230H In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2016-11-23 Classification: TRANSFERASE Ligands: CL, 62E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: CL, 62E
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Crystal Structure Of Cmet Wt With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2016-11-23 Classification: TRANSFERASE Ligands: 63B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: 63B
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Crystal Structure Of Cmet In Complex With Cmpd.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2016-11-23 Classification: TRANSFERASE Ligands: 63K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: 63K
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Crystal Structure Of C-Met L1195V In Complex With Sar125844
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2016-11-23 Classification: TRANSFERASE Ligands: 63K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: 63K
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Crystal Structure Of C-Met-M1250T In Complex With Sar125844.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-11-23 Classification: TRANSFERASE Ligands: 63K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: 63K
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Discovery Of (2S)-8-((3R)-3-Methylmorpholin-4-Yl)-1-(3-Methyl-2-Oxo- Butyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido(1,2-A)Pyrimidin-6- One: A Novel Potent And Selective Inhibitor Of Vps34 For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2014-11-26 Classification: TRANSFERASE Ligands: EUT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: EUT
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Discovery Of (2S)-8-((3R)-3-Methylmorpholin-4-Yl)-1-(3-Methyl-2-Oxo- Butyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido(1,2-A)Pyrimidin-6- One: A Novel Potent And Selective Inhibitor Of Vps34 For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2014-11-26 Classification: TRANSFERASE Ligands: SO4, RBQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: SO4, RBQ
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Discovery Of (2S)-8-((3R)-3-Methylmorpholin-4-Yl)-1-(3-Methyl-2-Oxo- Butyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido(1,2-A)Pyrimidin-6- One: A Novel Potent And Selective Inhibitor Of Vps34 For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2014-11-26 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
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Discovery Of (2S)-8-((3R)-3-Methylmorpholin-4-Yl)-1-(3-Methyl-2-Oxo- Butyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido(1,2-A)Pyrimidin-6- One: A Novel Potent And Selective Inhibitor Of Vps34 For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2014-11-26 Classification: TRANSFERASE Ligands: SO4, GOL, UJB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: SO4, GOL, UJB
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Discovery Of (2S)-8-((3R)-3-Methylmorpholin-4-Yl)-1-(3-Methyl-2-Oxo- Butyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido(1,2-A)Pyrimidin-6- One: A Novel Potent And Selective Inhibitor Of Vps34 For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-11-26 Classification: TRANSFERASE Ligands: SO4, 7A5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: SO4, 7A5
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Crystal Structure Of Vps34 In Complex With Sar405.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-10-22 Classification: LIPID KINASE Ligands: SO4, 1TT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-22
Ligands: SO4, 1TT
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Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2011-10-26 Classification: CHAPERONE Ligands: YK9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: YK9
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Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YJW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YJW
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Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YJX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YJX
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Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YJW, YJX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YJW, YJX
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Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YKB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YKB
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Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YKC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YKC
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Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YKE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YKE
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Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YKI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YKI
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Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YKJ
