Search Count: 12
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Salt-Inducible Kinase 3 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2024-01-10 Classification: SIGNALING PROTEIN Ligands: VRU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: VRU
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Crystal Structure Of The Catalytic Domain Of Adamts-5 In Complex With The Inhibitor Glpg1972
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2021-04-14 Classification: HYDROLASE Ligands: ZN, CA, OU5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: ZN, CA, OU5
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N-Terminal Bromodomain Of Human Brd2 With I-Bet726 (Gsk1324726A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-10-08 Classification: TRANSCRIPTION Ligands: EDO, 73B, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: EDO, 73B, SO4
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C-Terminal Bromodomain Of Human Brd2 With I-Bet726 (Gsk1324726A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-10-08 Classification: TRANSCRIPTION Ligands: 73B, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 73B, SO4
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N-Terminal Bromodomain Of Human Brd2 With 1-((2R,4S)-2-Methyl-4-(Phenylamino)-6-(4-(Piperidin-1-Ylmethyl)Phenyl)-3,4-Dihydroquinolin-1(2H)-Yl)Ethanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2014-10-08 Classification: TRANSCRIPTION Ligands: 9S3, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 9S3, SO4, DMS
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N-Terminal Bromodomain Of Human Brd4 With Gsk1324726A (I-Bet726)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2013-10-02 Classification: DNA BINDING PROTEIN Ligands: 73B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-02
Ligands: 73B
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Discovery Of Epigenetic Regulator I-Bet762: Lead Optimization To Afford A Clinical Candidate Inhibitor Of The Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2013-10-02 Classification: CELL CYCLE Ligands: H4C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-02
Ligands: H4C
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Discovery Of Epigenetic Regulator I-Bet762: Lead Optimization To Afford A Clinical Candidate Inhibitor Of The Bet Bromodomains
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2013-10-02 Classification: CELL CYCLE Ligands: L5S, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-02
Ligands: L5S, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd2 With The Inhibitor Gw841819X
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-06-15 Classification: NUCLEAR PROTEIN Ligands: WSH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: WSH, SO4
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Crystal Structure Of The First Bromodomain Of Human Brd2 With The Inhibitor Gsk525762 (Ibet)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2011-06-15 Classification: SIGNALING PROTEIN Ligands: EAM, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: EAM, SO4
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Crystal Structure Of The First Bromodomain Of Human Brd4 With The Inhibitor Gw841819X
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2011-06-15 Classification: SIGNALING PROTEIN Ligands: EDO, WSH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: EDO, WSH
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Crystal Structure Of The Second Bromodomain Of Human Brd4 With The Inhibitor Gw841819X
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-06-15 Classification: SIGNALING PROTEIN Ligands: WSH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: WSH
