Search Count: 14
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Identification Of Potent And Selective Ripk2 Inhibitors For The Treatment Of Inflammatory Diseases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2017-10-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 9WS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: 9WS, SO4
 |
Identification Of Potent And Selective Ripk2 Inhibitors For The Treatment Of Inflammatory Diseases.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2017-10-25 Classification: Transferase/Transferase Inhibitor Ligands: 9XA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: 9XA
 |
Egfr Kinase Domain In Complex With A Covalent Aminobenzimidazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2016-07-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5X4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-27
Ligands: 5X4
 |
Egfr Kinase Domain T790M Mutant In Complex With A Covalent Aminobenzimidazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-07-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5X4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-27
Ligands: 5X4
 |
Egfr Kinase Domain In Complex With A Covalent Aminobenzimidazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2016-07-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5XH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-27
Ligands: 5XH
 |
Cathepsin S In Complex With Non Covalent Arylaminoethyl Amide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2007-05-08 Classification: HYDROLASE Ligands: SO4, GNQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-05-08
Ligands: SO4, GNQ
 |
Crystal Structure Of Cathepsin S In Complex With A Zinc Mediated Non-Covalent Arylaminoethyl Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2006-08-15 Classification: HYDROLASE Ligands: ZN, CL, GNQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-15
Ligands: ZN, CL, GNQ
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A Dual Inhibitor Of The Leukocyte Proteases Cathepsin G And Chymase With Therapeutic Efficacy In Animals Models Of Inflammation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: NAG, SO4, CO, OHH, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: NAG, SO4, CO, OHH, MES
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A Dual Inhibitor Of The Leukocyte Proteases Cathepsin G And Chymase With Therapeutic Efficacy In Animals Models Of Inflammation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: SO4, OHH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: SO4, OHH
 |
Identification Of Novel Potent Bicyclic Peptide Deformylase Inhibitors
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2004-03-30 Classification: HYDROLASE Ligands: NI, GNR, GOL |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2004-03-30
Ligands: NI, GNR, GOL
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Potent, Small Molecule Inhibitors Of Human Mast Cell Tryptase. Anti-Asthmatic Action Of A Dipeptide-Based Transition State Analogue Containing Benzothiazole Ketone
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2003-09-23 Classification: HYDROLASE Ligands: CA, SO4, ABB |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2003-09-23
Ligands: CA, SO4, ABB
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Cathepsin-G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2002-05-01 Classification: HYDROLASE Ligands: KTP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-05-01
Ligands: KTP
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Thrombin Inhibitor From Theonalla, Cyclotheanamide-Based Macrocyclic Tripeptide Motif
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 1998-03-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1ZV |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1998-03-18
Ligands: 1ZV
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Molecular Basis For The Inhibition Of Human Alpha-Thrombin By The Macrocyclic Peptide Cyclotheonamide A
Organism: Homo sapiens, Theonella sp.
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1994-01-31 Classification: HYDROLASE/hydrolase inhibitor |
Organism: Homo sapiens, Theonella sp.
Method: X-RAY DIFFRACTION
Release Date: 1994-01-31