Search Count: 18
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Pdgfra-T674I In Complex With Covalent Ponatinib Derivative 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-02-12 Classification: TRANSFERASE Ligands: A1IRC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IRC
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C-Kit Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI, SO4
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 98A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 98A
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9XO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9XO
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9OO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9OO
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9VV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9VV
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: EDO, 9WU, BR, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: EDO, 9WU, BR, CL
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9KI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9KI
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C-Kit T670I Mutated Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI
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Pdgfra T674I Mutant Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI, PEG
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Pdgfra T674I Mutant Kinase Domain In Complex With Avapritinib Derivative 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9OO, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9OO, PEG
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Pdgfra Wild-Type Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2023-12-27 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
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Apo Crystal Structure Of Pdgfra-T674I Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-12-27 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor Borussertib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-03-20 Classification: TRANSFERASE Ligands: G4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-20
Ligands: G4K
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-02-20 Classification: TRANSFERASE Ligands: G4T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G4T
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 31
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-02-20 Classification: TRANSFERASE Ligands: G4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G4Q
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 30B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-02-20 Classification: TRANSFERASE Ligands: G4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G4N
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 24B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-02-20 Classification: TRANSFERASE Ligands: G4H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G4H
