Search Count: 21
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Structural Basis Of Impaired Hydrolysis In Kras Q61H Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2020-04-15 Classification: HYDROLASE Ligands: GTP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: GTP, MG
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Gdp-Bound Kras P34R Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2020-04-15 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: GDP, MG
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Kras P34R Mutant Structure In Complex With Gtp Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-04-15 Classification: HYDROLASE Ligands: GNP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: GNP, MG
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Crystal Structure Of Human Kras P34R Mutant In Complex With Gnp And Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-03-11 Classification: HYDROLASE Ligands: GNP, MG, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-11
Ligands: GNP, MG, PO4
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Crystal Structure Of Human Kras P34R Mutant In Complex With Gnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-02-26 Classification: HYDROLASE Ligands: MG, PO4, GNP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: MG, PO4, GNP
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Crystal Structure Of Kras V14I-Gdp Demonstrating Open Switch 1 Conformation - Form 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-07-31 Classification: HYDROLASE Ligands: GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GDP
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Crystal Structure Of Kras V14I-Gdp Demonstrating Disorder Switch 1 Conformation - Form 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-07-31 Classification: HYDROLASE Ligands: GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GDP
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Crystal Structure Of Kras A146T-Gdp Demonstrating Open Switch 1 Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2019-05-22 Classification: HYDROLASE Ligands: GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: GDP
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Src Kinase Bound To Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-02-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6H3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: 6H3
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Crystal Structure Of Erk2 Covalently Bound To Sm1-71
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: SO4, 6H3, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: SO4, 6H3, EDO, CL
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Crystal Structure Of Erk1 Covalently Bound To Sm1-71
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: 6H3, EWH, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: 6H3, EWH, SO4, EDO
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Kras Mutant-D33E In Gdp-Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2018-01-24 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-24
Ligands: GDP, MG
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Kras Mutant-A59G In Gdp-Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-01-24 Classification: HYDROLASE Ligands: MG, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-24
Ligands: MG, GDP
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Crystal Structure Of Human Kras A59G Mutant In Complex With Gcp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-01-24 Classification: HYDROLASE Ligands: GCP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-24
Ligands: GCP
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Kras G12C In Bound To Quinazoline Based Switch Ii Pocket (Swiip) Binder
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-08-23 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: GDP, MG, 8ZG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-23
Ligands: GDP, MG, 8ZG
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Covalent Gtp-Competitive Inhibitors Of Kras G12C: Guanosine Bisphosphonate Analogs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-04-12 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 6ZD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-12
Ligands: 6ZD
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Glutathione S-Transferase Bound With Hydrolyzed Piperlongumine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2016-11-30 Classification: transferase/transferase inhibitor Ligands: 3LF, GSH, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: 3LF, GSH, MES
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Crystal Structure Of A Gdp-Bound G12R Oncogenic Mutant Of Human Gtpase Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.04 Å Release Date: 2015-06-10 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: GDP, MG
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Crystal Structure Of A Gdp-Bound G12V Oncogenic Mutant Of Human Gtpase Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2015-06-10 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: GDP, MG
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Crystal Structure Of A Gdp-Bound G13D Oncogenic Mutant Of Human Gtpase Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2015-06-10 Classification: HYDROLASE Ligands: GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-10
Ligands: GDP, MG
