Search Count: 14
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Human Apo Hcn1 Nanodisc
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Resolution:2.50 Å Release Date: 2026-05-20 Classification: MEMBRANE PROTEIN |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2026-05-20
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Human Hcn1 In Complex With Camp In Nanodisc
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:2.60 Å Release Date: 2026-05-20 Classification: MEMBRANE PROTEIN Ligands: CMP |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-05-20
Ligands: CMP
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Crystal Structure Of The Unliganded Form Of Hcn2 Cnbd
Organism: Escherichia coli o157:h7, Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2016-11-30 Classification: TRANSPORT PROTEIN Ligands: NO3 |
Organism: Escherichia coli o157:h7, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2016-11-30
Ligands: NO3
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Itk Kinase Domain In Complex With Compound 1 N-{1-[(1,1-Dioxo-1-Thian-2-Yl)(Phenyl)Methyl]-1H- Pyrazol-4-Yl}-5,5-Difluoro-5A-Methyl-1H,4H,4Ah,5H,5Ah,6H-Cyclopropa[F]Indazole-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-04-29 Classification: TRANSFERASE/INHIBITOR Ligands: 3P6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-29
Ligands: 3P6
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Compound 21 (1-Alkyl-Substituted 1,2,4-Triazoles)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2013-01-09 Classification: Transferase/Transferase Inhibitor Ligands: 17V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-09
Ligands: 17V
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Rational Design Of Pi3K-Alpha Inhibitors That Exhibit Selectivity Over The Pi3K-Beta Isoform
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-11-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3T8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-16
Ligands: 3T8
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Discovery Of Gdc-0980: A Potent, Selective, And Orally Available Class I Phosphatidylinositol 3-Kinase (Pi3K)/Mammalian Target Of Rapamycin (Mtor) Kinase Inhibitor For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2011-11-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 980 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-02
Ligands: 980
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Structure-Based Design Of Thienobenzoxepin Inhibitors Of Pi3- Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-08-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FAV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-03
Ligands: FAV
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Structure-Based Design Of Thienobenzoxepin Inhibitors Of Pi3-Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2011-08-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FAZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-03
Ligands: FAZ
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Crystal Structures Of Pan-Pi3-Kinase And Dual Pan-Pi3-Kinase/Mtor Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2010-02-16 Classification: TRANSFERASE Ligands: JZW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: JZW
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Discovery Of (Thienopyrimidin-2-Yl)Aminopyrimidines As Potent, Selective, And Orally Available Pan-Pi3-Kinase And Dual Pan-Pi3-Kinase/Mtor Inhibitors For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2010-02-16 Classification: TRANSFERASE Ligands: JZX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: JZX
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Discovery Of (Thienopyrimidin-2-Yl)Aminopyrimidines As Potent, Selective, And Orally Available Pan-Pi3-Kinase And Dual Pan-Pi3-Kinase/Mtor Inhibitors For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2010-02-16 Classification: TRANSFERASE Ligands: JZY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: JZY
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Structural Model For The Fe-Containing Isoform Of Acireductone Dioxygenase
Organism: Klebsiella oxytoca
Method: SOLUTION NMR Release Date: 2006-10-24 Classification: OXIDOREDUCTASE Ligands: FE2 |
Organism: Klebsiella oxytoca
Method: SOLUTION NMR
Release Date: 2006-10-24
Ligands: FE2
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Short Factor Viia With A Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2005-01-18 Classification: HYDROLASE Ligands: CA, SO4, 905 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-01-18
Ligands: CA, SO4, 905
