Search Count: 31
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Receptor For Advanced Glycation End Products Vc1 Domain In Complex With 3-(3-(((3-(4-Carboxyphenoxy)Benzyl)Oxy)Methyl)Phenyl)-1H-Indole-2-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2021-12-15 Classification: SIGNALING PROTEIN Ligands: ACT, CL, Y6S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-15
Ligands: ACT, CL, Y6S
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Structure Of Tim-3 In Complex With 8-Chloro-2-Methyl-9-(3-Mehtylpyridin-4-Yl)-[1,2,4]Triazolo[1,5-C]Quinazolin-5(6H)-One (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2021-10-13 Classification: IMMUNE SYSTEM Ligands: YQ7, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: YQ7, CA
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Structure Of Tim-3 In Complex With N-(4-(8-Chloro-2-Mehtyl-5-Oxo-5,6-Dihydro-[1,2,4]Triazolo[1,5-C]Quinazolin-9-Yl)-3-Methylphenyl)Methanesulfonamdide (Compound 35)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2021-10-13 Classification: IMMUNE SYSTEM Ligands: YQD, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: YQD, CA
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Structure Of Tim-3 In Complex With N-(4-(8-Chloro-2-Methyl-5-Oxo-5,6-Dihydro-[1,2,4]Traizolo[1,5-C]Quinazolin-9-Yl)-3-Methylphenyl)-1H-Imidazole-2-Sulfonamide (Compound 38)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-10-13 Classification: IMMUNE SYSTEM Ligands: YQG, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: YQG, CA
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Receptor For Advanced Glycation End Products Vc1 Domain In Complex With 3-(3-((4-(4-Carboxyphenoxy)Benzyl)Oxy)Phenyl)-1H-Indole-2-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-07-28 Classification: SIGNALING PROTEIN Ligands: Y6P, ACT, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: Y6P, ACT, CL
 |
Receptor For Advanced Glycation End Products Vc1 Domain In Complex With 3-(3-((4-(4-Carboxyphenoxy)Benzyl)Oxy)Phenyl)-1H-Indole-2-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2021-07-14 Classification: SIGNALING PROTEIN Ligands: ACT, CL, V74 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ACT, CL, V74
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Receptor For Advanced Glycation End Products Vc1 Domain In Complex With 3-(3-(((3-(4-Carboxyphenoxy)Benzyl)Oxy)Methyl)Phenyl)-1H-Indole-2-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2021-07-14 Classification: SIGNALING PROTEIN Ligands: ACT, CL, V6Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ACT, CL, V6Y
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Receptor For Advanced Glycation End Products Vc1 Domain In Complex With Fragment 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-07-14 Classification: SIGNALING PROTEIN Ligands: ACT, CL, V6M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ACT, CL, V6M
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Receptor For Advanced Glycation End Products Vc1 Domain In Complex With Fragment 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2021-07-14 Classification: SIGNALING PROTEIN Ligands: ACT, CL, V6P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ACT, CL, V6P
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Receptor For Advanced Glycation End Products Vc1 Domain In Complex With Fragment 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-07-14 Classification: SIGNALING PROTEIN Ligands: ACT, V6V, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ACT, V6V, CL
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Receptor For Advanced Glycation End Products Vc1 Domain In Complex With Fragments 1 & 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2021-07-14 Classification: SIGNALING PROTEIN Ligands: ACT, V6M, V6P, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ACT, V6M, V6P, CL
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Receptor For Advanced Glycation End Products Vc1 Domain In Complex With Fragments 1 & 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-07-14 Classification: SIGNALING PROTEIN Ligands: ACT, V6S, V6M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ACT, V6S, V6M
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Discovery And Structure-Based Optimization Of Potent And Selective Wdr5 Inhibitors Containing A Dihydroisoquinolinone Bicyclic Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2020-01-01 Classification: TRANSCRIPTION Ligands: Q41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: Q41
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Wd Repeat-Containing Protein 5 Complexed With N-[(3,5-Dimethoxyphenyl)Methyl]-4'-Fluoro-5-{[(2E)-2-Imino-3-Methyl-2,3-Dihydro-1H-Imidazol-1-Yl]Methyl}-2'-Methyl[1,1'-Biphenyl]-3-Carboxamide (Compound 13)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2020-01-01 Classification: GENE REGULATION/INHIBITOR Ligands: Q6S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: Q6S
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Wdr5 In Complex With A Win Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-03-13 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HH7, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HH7, DMS, SO4
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Wdr5 In Complex With A Win Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2019-03-13 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HHM, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HHM, SO4, DMS
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Discovery Of Potent 2-Aryl-6,7-Dihydro-5Hpyrrolo[ 1,2-A]Imidazoles As Wdr5 Win-Site Inhibitors Using Fragment-Based Methods And Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLM
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLP
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLS, SO4
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLJ, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-13
Ligands: HLJ, EPE