Search Count: 9
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Discovery Of A Kras G12V Inhibitor In Vivo Tool Compound Starting From An Hsqc-Nmr Based Fragment Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-11-09 Classification: SIGNALING PROTEIN Ligands: 2XO, GDP, MG, LX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: 2XO, GDP, MG, LX6
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Crystal Structure Of Kras-G12C In Complex With Compound 23 (Bi-0474)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXD
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Crystal Structure Of Kras-G12C In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXK, SO4
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Crystal Structure Of Bit-Blocked Kras-G12V-S39C In Complex With Compound 20A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, 2XO, MG, LXU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, 2XO, MG, LXU
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Crystal Structure Of Compound 10 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IOD, IFJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IOD, IFJ
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Crystal Structure Of Compound 6 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IFF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IFF
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Crystal Structure Of Compound 4 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IF8, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IF8, ZN
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Crystal Structure Of Protac 5 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2022-09-07 Classification: LIGASE Ligands: IEI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-07
Ligands: IEI
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Crystal Structure Of Mdm2 In Complex With Compound 13.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2018-12-19 Classification: LIGASE Ligands: H28, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: H28, GOL, SO4